A new, one-pot, three-component synthesis of 4H-pyrido [1, 2-a] pyrimidines, 4H-pyrimido [1, 2-a] pyrimidines, and 4H-pyrazino [1, 2-a] pyrimidines

M Adib, MH Sayahi, H Ziyadi, HR Bijanzadeh, LG Zhu - Tetrahedron, 2007 - Elsevier
A new, one-pot and three-component synthesis of 4H-pyrido [1, 2-a] pyrimidines, 4H-
pyrimido [1, 2-a] pyrimidines, and 4H-pyrazino [1, 2-a] pyrimidines is described. The reactive …

A novel, one-pot, three-component synthesis of 4H-pyrido [1, 2-a] pyrimidines

M Adib, MH Sayahi, M Nosrati, LG Zhu - Tetrahedron letters, 2007 - Elsevier
A novel, one-pot, three-component synthesis of 4H-pyrido [1, 2-a] pyrimidines is described.
The reactive 1: 1 zwitterionic intermediate, formed by the addition of isocyanides to dialkyl …

New efficient approach for the synthesis of 2‐alkyl(aryl) substituted 4H‐pyrido[1,2‐a]pyrimidin‐4‐ones

HG Bonacorso, FJ Righi, IR Rodrigues… - Journal of …, 2006 - Wiley Online Library
A new, efficient and easy route for the preparation of a series of 2‐alkyl (aryl) substituted 4‐
oxo‐4H‐pyrido‐[1, 2‐a] pyrimidines, where alkyl= CH3; aryl= C6H5, 4‐FC6H4, 4‐ClC6H4, 4 …

Efficient synthesis of novel pyrano [2, 3-d] pyrido [1, 2-a] pyrimidine derivatives via isocyanide-based three-component reactions

AA Esmaeili, F Salehan, A Habibi, AR Fakhari - Tetrahedron Letters, 2016 - Elsevier
The synthesis of novel tricyclic fused pyrano [2, 3-d] pyrido [1, 2-a] pyrimidines containing
both biologically active pyridopyrimidine and pyranopyrimidine scaffolds, via the reaction of …

Synthesis of 3,4-Dihydropyridin-2(1H)-ones and 3,4-Dihydro-2H-pyrans via Four-Component Reactions of Aromatic Aldehydes, Cyclic 1,3-Carbonyls, Arylamines …

J Sun, EY Xia, Q Wu, CG Yan - ACS Combinatorial Science, 2011 - ACS Publications
A protocol has been developed for the efficient synthesis of structurally diverse 3, 4-
dihydropyridin-2 (1 H)-ones and 3, 4-dihydro-2 H-pyrans via four-component reactions of …

A novel four component one-pot access to pyrindines and tetrahydroquinolines

NAM Yehia, K Polborn, TJJ Müller - Tetrahedron letters, 2002 - Elsevier
Dihydropyrindines and tetrahydroquinolines, ie cyclopentyl and cyclohexyl annealed
pyridines, can be synthesized in good yields in a one-pot three-step four-component …

A convenient, one step synthesis of pyrano [2, 3-b] pyridines

N Martin, C Seoane, JL Soto - Tetrahedron, 1988 - Elsevier
A novel, one step synthesis of pyrano [2, 3-b] pyri-dines from malononitrile and unsaturated
ketones is reported. The reaction mechanism is discussed and takes place through an …

Tetrahydropyridinium bromide: Useful synthon to functionalized pyrrolidines

L Guideri, R Noschese… - Journal of Heterocyclic …, 2012 - Wiley Online Library
benzyl‐5‐(ethoxycarbonyl)‐2, 3, 4, 5‐tetrahydropyridinium bromide undergoes ring
contraction with a series of nucleophiles, getting 2, 2‐disubstitued pyrrolidines. Moreover …

Efficient Synthesis of Highly Functionalized Dihydropyrido[2,3-d]pyrimidines by a Double Annulation Strategy from α-Alkenoyl-α-carbamoyl Ketene-(S,S)-acetals

L Zhao, F Liang, X Bi, S Sun, Q Liu - The Journal of Organic …, 2006 - ACS Publications
A convenient and efficient synthesis of highly functionalized dihydropyrido [2, 3-d]
pyrimidines via a double [5+ 1] annulation strategy starting from easily available α-alkenoyl …

[PDF][PDF] Novel syntheses of pyrido [1, 2-a] pyrimidin-2-ones, 2H-quinolizin-2-ones, pyrido [1, 2-a] quinolin-3-ones, and thiazolo [3, 2-a] pyrimidin-7-ones

AR Katritzky, JW Rogers, RM Witek, SK Nair - Arkivoc, 2004 - arkat-usa.org
Abstract As novel 1, 3-bis-electrophilic synthons, 1-benzotriazolyl-2-propynones provide
access to the fused ring systems of pyrido [1, 2-a] pyrimidin-2-ones and 2H-quinolizin-2 …