Cationic and Anionic Requirements for the Binding of 2β‐Carbomethoxy‐3β‐(4‐Fluorophenyl)[3H]tropane to the Dopamine Uptake Carrier
MEA Reith, LL Coffey - Journal of neurochemistry, 1993 - Wiley Online Library
The present study reports the ion dependency of 2β‐carbomethoxy‐3β‐(4‐fluorophenyl)[3H]
tropane ([3H]‐CFT) binding to the dopamine transporter in the rat striaturn. The results …
tropane ([3H]‐CFT) binding to the dopamine transporter in the rat striaturn. The results …
Methyl 3β‐(4‐[125I]Iodophenyl)Tropane‐2β‐Carboxylate In Vitro Binding to Dopamine and Serotonin Transporters Under “Physiological” Conditions
M Laruelle, SS Giddings, Y Zea‐Ponce… - Journal of …, 1994 - Wiley Online Library
Methyl 3β‐(4‐[125I] iodophenyl) tropane‐2β‐carboxylate ([123I] β‐CIT) is a single photon
emission computed tomographic radiotracer for in vivo labeling of dopamine (DA) and …
emission computed tomographic radiotracer for in vivo labeling of dopamine (DA) and …
Cationic interactions at the human dopamine transporter reveal binding conformations for dopamine distinguishable from those for the cocaine analog 2α …
N Chen, LL Sun, MEA Reith - Journal of neurochemistry, 2002 - Wiley Online Library
In membrane preparations, CFT, a phenyltropane cocaine analog, and dopamine (DA)
interact with the recombinant human dopamine transporter (hDAT) in Na+‐free medium …
interact with the recombinant human dopamine transporter (hDAT) in Na+‐free medium …
Translocation of dopamine and binding of 2β-carbomethoxy-3 β-(4-fluorophenyl) tropane (WIN 35,428) measured under identical conditions in rat striatal …
C Xu, LL Coffey, MEA Reith - Biochemical pharmacology, 1995 - Elsevier
Translocation of [3H] dopamine and binding of 2 β-carbomethoxy-3 β-(4-fluorophenyl)[3H]-
tropane ([3H] WIN 35,428) were measured in crude synaptosomal preparations from rat …
tropane ([3H] WIN 35,428) were measured in crude synaptosomal preparations from rat …
Characterization of a tropane radioligand,[3H] 2β-Propanoyl-3β-(4-tolyl) Tropane ([3H] PTT), for dopamine transport sites in rat brain
SR Letchworth, HR Smith, LJ Porrino, BA Bennett… - … of Pharmacology and …, 2000 - ASPET
PTT (2β-propanoyl-3β-[4-tolyl] tropane) is a tropane analog relatively selective for dopamine
transporters in binding and uptake assays in vitro, with long-acting psychostimulant …
transporters in binding and uptake assays in vitro, with long-acting psychostimulant …
Modeling of the pH dependence of the binding of WIN 35,428 to the dopamine transporter in rat striatal membranes: is the bioactive form positively charged or neutral?
C Xu, ME Reith - Journal of Pharmacology and Experimental …, 1996 - ASPET
Cocaine and its phenyltropane analogs, including 2beta-carbomethoxy-3beta-(4-
fluorophenyl) tropane can exist in either the cationic or the neutral form, with the proportion …
fluorophenyl) tropane can exist in either the cationic or the neutral form, with the proportion …
[PDF][PDF] Binding of the cocaine analog 2 beta-carbomethoxy-3 beta-(4-[125I] iodophenyl) tropane to serotonin and dopamine transporters: different ionic requirements …
SUMMARY The iodinated cocaine analog 2/3-carbomethoxy-3fl-(4-[125l] iodophenyl)
tropane(j9-[125l} CIT) binds with high affinity to the platelet plasma membrane serotonin …
tropane(j9-[125l} CIT) binds with high affinity to the platelet plasma membrane serotonin …
N-(3-iodoprop-2E-enyl)-2β-Carbomethoxy-3β-(3′, 4′-dichlorophenyl) nortropane (β-CDIT), a tropane derivative: Pharmacological characterization as a specific …
N-(3-Iodoprop-2 E-enyl)-2β-carbomethoxy-3β-(3′, 4′-dichlorophenyl) nortropane (β-
CDIT), a new iodinated tropane derivative, has been synthesized and radiolabeled with …
CDIT), a new iodinated tropane derivative, has been synthesized and radiolabeled with …
Modeling of the Interaction of Na+ and K+ with the Binding of the Cocaine Analogue 3β‐(4‐[125I]Iodophenyl)tropane‐2β‐Carboxylic Acid Isopropyl Ester to the …
NH Chen, JH Ding, YL Wang… - Journal of …, 1997 - Wiley Online Library
The present study examines the interaction of Na+ and K+ with the binding of the cocaine
analogue 3β‐(4‐[125I] iodophenyl) tropane‐2β‐carboxylic acid isopropyl ester to dopamine …
analogue 3β‐(4‐[125I] iodophenyl) tropane‐2β‐carboxylic acid isopropyl ester to dopamine …
Binding of the [125I]3β‐(Iodophenyl)tropan‐2β‐carboxylic acid isopropyl ester to the dopamine transporter at a physiologically relevant temperature: Mutually …
NH Chen, YL Wang, MEA Reith - Synapse, 1997 - Wiley Online Library
The present study describes the binding of cocaine analog [125I] 3β‐(iodophenyl) tropan‐2β‐
carboxylic acid isopropyl ester ([125I] RTI‐121), a highly selective ligand for the dopamine …
carboxylic acid isopropyl ester ([125I] RTI‐121), a highly selective ligand for the dopamine …
相关搜索
- tropane 2β dopamine transporter
- win 35,428 dopamine transporter
- modeling of the interaction dopamine transporter
- isopropyl ester dopamine transporter
- tropane 2β physiological conditions
- tropane 2β modeling of the interaction
- tropane 2β isopropyl ester
- cationic interactions binding conformations
- rat brain propanoyl 3β