8‐Hydroxyquinoline‐2‐Carboxanilides as antiviral agents against avian influenza virus

J Kos, CF Ku, I Kapustikova, M Oravec… - …, 2019 - Wiley Online Library
Abstract Series of thirty‐two mono‐, di‐and tri‐substituted 8‐hydroxyquinoline‐2‐
carboxanilides were prepared by microwave‐assisted synthesis. The compounds were …

Novel 3-sulphonamido-quinazolin-4(3H)-One Derivatives: Microwave-Assisted Synthesis and Evaluation of Antiviral Activities against Respiratory and Biodefense …

P Selvam, P Vijayalakshimi, DF Smee… - Antiviral Chemistry …, 2007 - journals.sagepub.com
We designed and synthesized novel 2, 3-disubstituted quinazolin-4 (3 H)-ones by
microwave technique and characterized them by spectral analysis. Synthesized compounds …

Heterocyclic compounds based on 3-(4-bromophenyl) azo-5-phenyl-2 (3H)-furanone: Anti-avian influenza virus (H5N1) activity

EM Flefel, RE Abdel-Mageid, WA Tantawy, MA Ali… - Acta …, 2012 - hrcak.srce.hr
Sažetak 3-[2-(4-Bromphenyl) hydrazono]-5-phenyl-furan-2 (3H)-one (1) was used for
preparation of some novel pyrazole, pyridazinone, oxadiazole, triazole, thiazolidine and …

Antiviral activity of amides and carboxamides of quinolizidine alkaloid (−)-cytisine against human influenza virus A (H1N1) and parainfluenza virus type 3

VA Fedorova, RA Kadyrova, AV Slita… - Natural product …, 2021 - Taylor & Francis
Novel derivatives of quinolizidine alkaloid (−)-cytisine were synthesised. ADME properties,
cytotoxicity against HEK293 cells and activity against viruses of influenza A/California/07/09 …

Synthesis and biological evaluation of 2‐oxo‐pyrazine‐3‐carboxamide‐yl nucleoside analogues and their epimers as inhibitors of influenza A viruses

J Gao, X Luo, Y Li, R Gao, H Chen… - Chemical Biology & Drug …, 2015 - Wiley Online Library
Novel 2‐oxo‐pyrazine‐3‐carboxamide‐yl nucleoside analogues and their epimers were
designed, synthesized and evaluated for their activities against influenza A viruses H1N1 …

Ring-substituted 8-hydroxyquinoline-2-carboxanilides as potential antimycobacterial agents

J Kos, I Zadrazilova, E Nevin, M Soral, T Gonec… - Bioorganic & Medicinal …, 2015 - Elsevier
In this study, a series of twenty-two ring-substituted 8-hydroxyquinoline-2-carboxanilides
was prepared and characterized. Primary in vitro screening of the synthesized compounds …

Synthesis and evaluation for biological activity of 3-alkyl and 3-halogenoalkyl-quinoxalin-2-ones variously substituted. Part 4

A Carta, P Sanna, M Loriga, MG Setzu, P La Colla… - Il Farmaco, 2002 - Elsevier
A new series of 3-isopropyl-, 3-trifluoromethyl-and 3-bromomethylquinoxaline-2-ones
variously substituted on the benzo-moiety were synthesized and submitted to a preliminary …

Synthesis and Antiviral Bioactivity of Novel 3-((2-((1E,4E)-3-Oxo-5-arylpenta-1,4-dien-1-yl)phenoxy)methyl)-4(3H)-quinazolinone Derivatives

J Ma, P Li, X Li, Q Shi, Z Wan, D Hu… - Journal of agricultural …, 2014 - ACS Publications
A series of novel 3-((2-((1 E, 4 E)-3-oxo-5-arylpenta-1, 4-dien-1-yl) phenoxy) methyl)-4 (3 H)-
quinazolinone derivatives were designed and synthesized. Antiviral bioassays indicated that …

Synthesis, antiviral activity and cytotoxicity evaluation of Schiff bases of some 2-phenyl quinazoline-4 (3) H-ones

KS Kumar, S Ganguly, R Veerasamy… - European journal of …, 2010 - Elsevier
A new series of 3-(benzylideneamino)-2-phenylquinazoline-4 (3H)-ones were prepared
through Schiff base formation of 3-amino-2-phenyl quinazoline-4 (3) H-one with various …

Microwave assisted synthesis and anti-influenza virus activity of 1-adamantyl substituted N-(1-thia-4-azaspiro [4.5] decan-4-yl) carboxamide derivatives

F Göktaş, E Vanderlinden, L Naesens, N Cesur… - Bioorganic & medicinal …, 2012 - Elsevier
A microwave-assisted three-component one-pot cyclocondensation method was applied for
the synthesis of novel N-(1-thia-4-azaspiro [4.5] decan-4-yl) carboxamide compounds …