2-Phenylbenzofuran derivatives as butyrylcholinesterase inhibitors: synthesis, biological activity and molecular modeling
A series of 2-phenylbenzofurans compounds was designed, synthesized and evaluated as
cholinesterase inhibitors. The biological assay experiments showed that most of the …
cholinesterase inhibitors. The biological assay experiments showed that most of the …
1H-benzimidazole derivatives as butyrylcholinesterase inhibitors: synthesis and molecular modeling studies
G Coban, L Carlino, AH Tarikogullari, S Parlar… - Medicinal Chemistry …, 2016 - Springer
Abstract A series of N-{2-[2-(1 H-benzimidazole-2-yl) phenoxy] ethyl} substituted amine
derivatives were synthesized and tested for their cholinesterase inhibitor activity …
derivatives were synthesized and tested for their cholinesterase inhibitor activity …
Synthesis, biological activity and molecular modeling studies on 1H-benzimidazole derivatives as acetylcholinesterase inhibitors
AS Alpan, S Parlar, L Carlino, AH Tarikogullari… - Bioorganic & medicinal …, 2013 - Elsevier
Abstract A series of N-{2-[4-(1H-benzimidazole-2-yl) phenoxy] ethyl} substituted amine
derivatives were designed to assess cholinesterase inhibitor activities. Acetylcholinesterase …
derivatives were designed to assess cholinesterase inhibitor activities. Acetylcholinesterase …
2-Benzoyl-6-benzylidenecyclohexanone analogs as potent dual inhibitors of acetylcholinesterase and butyrylcholinesterase
In the present study, a series of 2-benzoyl-6-benzylidenecyclohexanone analogs have been
synthesized and evaluated for their anti-cholinesterase activity. Among the forty-one …
synthesized and evaluated for their anti-cholinesterase activity. Among the forty-one …
In silico studies on 2, 3-dihydro-1, 5-benzothiazepines as cholinesterase inhibitors
FL Ansari, S Kalsoom, Z Ali, F Jabeen - Medicinal Chemistry Research, 2012 - Springer
In vitro studies on cholinesterase inhibitory potential on the three sets of 2, 3-dihydro-1, 5-
benzothiazepines have been carried out. The compounds in Set 1 were unsubstituted on …
benzothiazepines have been carried out. The compounds in Set 1 were unsubstituted on …
Novel N-benzylpyridinium moiety linked to arylisoxazole derivatives as selective butyrylcholinesterase inhibitors: synthesis, biological evaluation, and docking study
F Vafadarnejad, E Karimpour-Razkenari, B Sameem… - Bioorganic …, 2019 - Elsevier
A novel series of N-benzylpyridinium moiety linked to arylisoxazole ring were designed,
synthesized, and evaluated for their in vitro acetylcholinesterase (AChE) and …
synthesized, and evaluated for their in vitro acetylcholinesterase (AChE) and …
Synthesis of 4-[(diethylamino) methyl]-phenol derivatives as novel cholinesterase inhibitors with selectivity towards butyrylcholinesterase
L Yu, R Cao, W Yi, Q Yan, Z Chen, L Ma… - Bioorganic & medicinal …, 2010 - Elsevier
A series of novel cholinesterase inhibitors, being composed of 4-[(diethylamino) methyl]-
phenoxy and secondary amine which were linked with a different length alkyl chain, were …
phenoxy and secondary amine which were linked with a different length alkyl chain, were …
Design, synthesis and bioactivity of novel phthalimide derivatives as acetylcholinesterase inhibitors
W Si, T Zhang, L Zhang, X Mei, M Dong… - Bioorganic & Medicinal …, 2016 - Elsevier
A series of novel phthalimide derivatives related to benzylpiperazine were synthesized and
evaluated as cholinesterase inhibitors. The results showed that all compounds were able to …
evaluated as cholinesterase inhibitors. The results showed that all compounds were able to …
Synthesis, characterization, and molecular docking analysis of novel benzimidazole derivatives as cholinesterase inhibitors
Two series of novel acetylcholinesterase (AChE) and butyrylcholinesterase (BChE)
inhibitors containing benzimidazole core structure were synthesized by a four-step reaction …
inhibitors containing benzimidazole core structure were synthesized by a four-step reaction …
Novel arylcarbamate-N-acylhydrazones derivatives as promising BuChE inhibitors: Design, synthesis, molecular modeling and biological evaluation
DAS Yamazaki, AMF Rozada, P Barea, EC Reis… - Bioorganic & Medicinal …, 2021 - Elsevier
A novel series of arylcarbamate-N-acylhydrazones derivatives have been designed and
synthesized as potential anti-cholinesterase agents. In vitro studies revealed that these …
synthesized as potential anti-cholinesterase agents. In vitro studies revealed that these …
相关搜索
- butyrylcholinesterase inhibitors molecular modeling
- butyrylcholinesterase inhibitors biological activity
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- acetylcholinesterase inhibitors phthalimide derivatives
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- buche inhibitors biological evaluation
- benzimidazole derivatives cholinesterase inhibitors
- butyrylcholinesterase inhibitors biological evaluation
- acetylcholinesterase inhibitors biological activity
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- molecular modeling biological evaluation