Oxidative furan-to-indole rearrangement. Synthesis of 2-(2-acylvinyl) indoles and flinderole C analogues
AS Makarov, AA Merkushev, MG Uchuskin… - Organic …, 2016 - ACS Publications
Oxidative rearrangement of 2-(2-aminobenzyl) furans affording 2-(2-acylvinyl) indoles in a
stereocontrolled manner in good-to-excellent yields has been developed. Thus,(2 …
stereocontrolled manner in good-to-excellent yields has been developed. Thus,(2 …
Furan ring opening–indole ring closure: recyclization of 2-(2-aminophenyl) furans into 2-(2-oxoalkyl) indoles
AS Pilipenko, VV Mel'chin, IV Trushkov, DA Cheshkov… - Tetrahedron, 2012 - Elsevier
The acid-catalyzed rearrangement of 5-alkyl-2-[2-(sulfonylamino) phenyl] furans into 2-(2-
oxoalkyl) indoles is described. When the N-sulfonyl group in the starting compounds was …
oxoalkyl) indoles is described. When the N-sulfonyl group in the starting compounds was …
A short total synthesis of the antimalarial flindersial alkaloids
A short, efficient and novel approach for the syntheses of bis‐indole alkaloids flinderoles A−
C, and desmethylflinderole C, is being described. The synthesis utilizes the optimized …
C, and desmethylflinderole C, is being described. The synthesis utilizes the optimized …
Furan as a 1, 3-diketone equivalent: the second type furan recyclization applied to indole synthesis
AV Butin - Tetrahedron letters, 2006 - Elsevier
Furan as a 1,3-diketone equivalent: the second type furan recyclization applied to indole
synthesis - ScienceDirect Skip to main contentSkip to article Elsevier logo Journals & Books …
synthesis - ScienceDirect Skip to main contentSkip to article Elsevier logo Journals & Books …
Furan ring opening—indole ring closure: pseudooxidative furan ring opening in the synthesis of indoles
AV Butin, SK Smirnov - Tetrahedron letters, 2005 - Elsevier
A new approach to the synthesis of 4-(2-indolyl)-3-buten-2-ones is described based on
condensation of 2-tosylaminobenzyl alcohols with N-tosylfurfurylamine. Pseudooxidative …
condensation of 2-tosylaminobenzyl alcohols with N-tosylfurfurylamine. Pseudooxidative …
Hydroxyalkylation of 4, 5, 6, 7-tetrahydroindole with polyfluorocarbonyl compounds as a route to 2-substituted indoles
AL Sigan, DV Gusev, ND Chkanikov, EY Shmidt… - Tetrahedron letters, 2011 - Elsevier
The regioselective hydroxyalkylation of 4, 5, 6, 7-tetrahydroindole at position 2 using highly
electrophilic polyfluorocarbonyl compounds was performed for the first time. Oxidation of the …
electrophilic polyfluorocarbonyl compounds was performed for the first time. Oxidation of the …
Facile synthesis of 6-hydroxyindole and 6-methoxyindole via regioselective Friedel-Crafts acylation and Baeyer-Villiger Oxidation
K Teranishi, S Nakatsuka, T Goto - synthesis, 1994 - thieme-connect.com
A facile synthesis of 6-hydroxyindole and 6-methoxyindole starting from indole is described.
Regioselective chloroacetylation of 1-pivaloylindole followed by Baeyer-Villiger oxidation …
Regioselective chloroacetylation of 1-pivaloylindole followed by Baeyer-Villiger oxidation …
Synthesis of spiro[2H‐indole‐2,1′‐1H‐isoindole]‐3,3′‐diones, spiro[1H‐isobenzofuran‐1,2′‐2H‐indole]‐3,3′‐diones and spiro[benzofuran‐2,1′‐isobenzofuran]‐3,3 …
JL Bullington, JH Dodd - Journal of heterocyclic chemistry, 1998 - Wiley Online Library
An auto oxidation‐rearrangement product 4 was isolated from a high dilution reaction of
ninhydrin with 3, 4, 5‐trimethoxyaniline in water. A general synthesis of this compound and …
ninhydrin with 3, 4, 5‐trimethoxyaniline in water. A general synthesis of this compound and …
A concise synthesis of 3-hydroxyindole-2-carboxylates by a modified Baeyer–Villiger oxidation
ZL Hickman, CF Sturino, N Lachance - Tetrahedron Letters, 2000 - Elsevier
A concise synthesis of 3-hydroxyindole-2-carboxylates by a modified Baeyer–Villiger
oxidation - ScienceDirect Skip to main contentSkip to article Elsevier logo Journals & Books …
oxidation - ScienceDirect Skip to main contentSkip to article Elsevier logo Journals & Books …
A straightforward synthesis of indole and benzofuran derivatives
V Fiandanese, D Bottalico, G Marchese, A Punzi - Tetrahedron, 2008 - Elsevier
A new methodology for the synthesis of indole and benzofuran derivatives has been
devised. The starting materials, ortho-substituted aryl diynes, have been easily converted …
devised. The starting materials, ortho-substituted aryl diynes, have been easily converted …