Characterisation of gestodene binding to the oestrogen receptor in human malignant breast tissue.

MJ Iqbal, AA Colletta - Anticancer Research, 1987 - europepmc.org
Gestodene, a new synthetic progestogen, binds to progesterone receptor (PR) derived from
normal breast, endometrium and both normal and diseased liver with an affinity 8-10 times …

A 12-month clinical investigation with a 24-day regimen containing 15 μg ethinylestradiol plus 60 μg gestodene with respect to hemostasis and cycle control

F Fruzzetti, AR Genazzani, C Ricci, F De Negri, C Bersi… - Contraception, 2001 - Elsevier
The effects of a 24-day regimen containing 15 μg ethinyl estradiol (EE) plus 60 μg
gestodene on cycle control and on hemostasis, were evaluated in 58 healthy women (age …

The oestrogenic effects of gestodene, a potent contraceptive progestin, are mediated by its A-ring reduced metabolites

AE Lemus, V Zaga, R Santillán… - Journal of …, 2000 - joe.bioscientifica.com
Gestodene (17 alpha-ethynyl-13 beta-ethyl-17 beta-hydroxy-4, 15-gonadien-3-one) is the
most potent synthetic progestin currently available and it is widely used as a fertility …

Intra-and interindividual variations in contraceptive steroid levels during 12 treatment cycles: no relation to irregular bleedings

C Jung-Hoffmann, H Kuhl - Contraception, 1990 - Elsevier
During one year of treatment with oral contraceptives containing 30 μg ethinylestradiol and
150 μg desogestrel (EE DG) or 30 μg EE and 75 μg gestodene (EE GSD), the serum …

[HTML][HTML] Effect of 21-day and 24-day oral contraceptive regimens containing gestodene (60 μg) and ethinyl estradiol (15 μg) on ovarian activity

H Sullivan, H Furniss, J Spona, M Elstein - Fertility and sterility, 1999 - Elsevier
Objective: To compare ovulation inhibition and ovarian activity with 21-day and 24-day
regimens of a low-dose combined oral contraceptive (COC) containing 60 μg of gestodene …

The safety and contraceptive efficacy of a 24-day low-dose oral contraceptive regimen containing gestodene 60 µg and ethinylestradiol 15 µg

Gestodene Study Group 322 - The European Journal of …, 1999 - Taylor & Francis
Objectives: The safety and contraceptive efficacy of a new 24-day regimen of an oral
contraceptive combination containing gestodene (GTD) 60 µg and ethinylestradiol (EE) 15 …

Influence of changes in the concentration of sex hormone-binding globulin in human serum on the protein binding of the contraceptive steroids levonorgestrel, 3-keto …

W Kuhnz, B Schütt, R Woloszczak - The Journal of Steroid Biochemistry …, 1994 - Elsevier
The serum protein binding of levonorgestrel, gestodene and 3-keto-desogestrel has been
determined during several clinical studies with different oral contraceptive formulations and …

Effect of troglitazone on the pharmacokinetics of an oral contraceptive agent

CM Loi, R Stern, JR Koup, AB Vassos… - The Journal of …, 1999 - Wiley Online Library
Fifteen healthy women participated in a study to determine the effect of multiple doses of
troglitazone on the pharmacokinetics of Ortho‐Novum 1/35 (35 μg ethinyl estradiol [EE] and …

A double-blind comparative study of the effects of a 23-day oral contraceptive regimen with 20 μg ethinyl estradiol and 75 μg gestodene and a 21-day regimen with 30 …

J Endrikat, C Klipping, C Gerlinger, A Ruebig… - Contraception, 2001 - Elsevier
In this double-blind study we compared the influence of two oral contraceptives, a 23-day
regimen with 20 μg ethinyl estradiol and 75 μg gestodene (23-day 20/75) and a 21-day …

Gestodene: a review of its pharmacology, potency and tolerability in combined contraceptive preparations

FZ Stanczyk, DF Archer - Contraception, 2014 - Elsevier
Combined progestin–estrogen pills are an established and reliable contraceptive option
used by women worldwide. Combined oral contraceptives (COCs) containing the progestins …