Pyrazoloquinazolinones and pyrazolopyridopyrimidinones by a sequential N-acylation–SNAr reaction

KK Gnanasekaran, NP Muddala, RA Bunce - Tetrahedron letters, 2015 - Elsevier
An efficient synthesis of pyrazolo [1, 5-a] quinazolin-5 (4H)-ones and pyrazolo [1, 5-a] pyrido
[3, 2-e] pyrimidin-5 (4H)-ones is reported from the reaction of 2-haloaroyl chlorides with 5 …

A new route for the synthesis of 1, 3, 4-trisubstituted pyrazolo [4, 3-c] quinolines via a multicomponent reaction

A Alizadeh, L Moafi, R Ghanbaripour, MH Abadi, Z Zhu… - Tetrahedron, 2015 - Elsevier
An efficient synthesis of a series of pyrazolo [4, 3-c] quinoline is reported. A multicomponent
reaction was designed using isatins, 1-aryl-2-(1, 1, 1-triphenyl-λ 5-phosphanylidene)-1 …

ZnCl2‐Promoted One‐Pot Three‐Component Synthesis of Multisubstituted Thiazolo[4,5‐b]pyridines and Thieno[2,3‐b:4,5‐b′]dipyridines

L Luo, L Meng, Y Peng, Y Xing, Q Sun… - European Journal of …, 2015 - Wiley Online Library
A ZnCl2‐promoted one‐pot synthesis of multisubstituted thiazolo [4, 5‐b] pyridines and
thieno [2, 3‐b: 4, 5‐b′] dipyridines from mercaptonitrile salts, α‐bromo ketones and ketones …

High Throughput Synthesis of Extended Pyrazolo[3,4-d]dihydropyrimidines

SV Ryabukhin, DS Granat, AS Plaskon… - ACS Combinatorial …, 2012 - ACS Publications
Thirteen 5-hetarylaminopyrazoles were synthesized in 62–93% yield through the arylation of
1-isopropyl-and 1-phenyl-5-aminopyrazoles with electrophilic hetarylhalides under …

Synthesis of spiro[pyrazolo[3,4-b] pyridine-4,3′-indoline] and spiro [benzo[h]pyrazolo[3,4-b]quinoline-4,3′-indoline] derivatives using wet cyanuric chloride under …

Z Yin, L Yang, L Wu - Journal of Chemical Sciences, 2013 - Springer
A simple and efficient synthesis of spiro [pyrazolo [3, 4-b] pyridine-4, 3′-indoline] and spiro
[benzo [h] pyrazolo [3, 4-b] quinoline-4, 3′-indoline] derivatives has been accomplished by …

Rapid synthesis of tetrahydroquinolines by indium trichloride catalyzed mono-and bis-intramolecular imino Diels–Alder reactions

RDRS Manian, J Jayashankaran, R Ramesh… - Tetrahedron letters, 2006 - Elsevier
A rapid synthesis of mono-and bis-tetrahydropyrazolo [4′, 3′: 5, 6] thiopyrano [4, 3-b]
quinolines has been achieved by the reaction of aldimines derived from aromatic amines …

3-Formylpyrazolo[1,5-a]pyrimidines as Key Intermediates for the Preparation of Functional Fluorophores

JC Castillo, A Tigreros, J Portilla - The Journal of Organic …, 2018 - ACS Publications
A one-pot route for the regioselective synthesis of 3-formylpyrazolo [1, 5-a] pyrimidines 4a–k
in good yields through a microwave-assisted process is provided. The synthesis proceeds …

[引用][C] New one‐step synthesis of pyrazolo[1,5‐a]pyrimidine and pyrazolo[1,5‐a]quinazoline derivatives via multicomponent reactions

BK Ghotekar, MN Jachak… - Journal of Heterocyclic …, 2009 - Wiley Online Library
A series of pyrazolopyrimidine and pyrazoloquinozoline derivatives has been synthesized in
one step by multicomponent reactions using, 5‐aminopyrazole, p …

A facile environment-friendly one-pot two-step regioselective synthetic strategy for 3,7-diarylpyrazolo[1,5-a]pyrimidines related to zaleplon and 3,6-diarylpyrazolo[1,5-a] …

AS Devi, S Kaping, JN Vishwakarma - Molecular diversity, 2015 - Springer
Aminopyrazoles required for the synthesis of pyrazolo 1, 5-a pyrimidines were obtained by
the reaction of enaminonitriles with hydrazine hydrate. The resulting aminopyrazoles are …

Recent synthetic methodologies for pyrazolo[1,5-a]pyrimidine

MA Salem, MH Helal, MA Gouda… - Synthetic …, 2019 - Taylor & Francis
The development of new synthetic routes towards pyrazolo [1, 5-a] pyrimidines for their
biological and medicinal exploration is an attractive area for researchers. This review …