Pyrazoloquinazolinones and pyrazolopyridopyrimidinones by a sequential N-acylation–SNAr reaction
KK Gnanasekaran, NP Muddala, RA Bunce - Tetrahedron letters, 2015 - Elsevier
An efficient synthesis of pyrazolo [1, 5-a] quinazolin-5 (4H)-ones and pyrazolo [1, 5-a] pyrido
[3, 2-e] pyrimidin-5 (4H)-ones is reported from the reaction of 2-haloaroyl chlorides with 5 …
[3, 2-e] pyrimidin-5 (4H)-ones is reported from the reaction of 2-haloaroyl chlorides with 5 …
A new route for the synthesis of 1, 3, 4-trisubstituted pyrazolo [4, 3-c] quinolines via a multicomponent reaction
An efficient synthesis of a series of pyrazolo [4, 3-c] quinoline is reported. A multicomponent
reaction was designed using isatins, 1-aryl-2-(1, 1, 1-triphenyl-λ 5-phosphanylidene)-1 …
reaction was designed using isatins, 1-aryl-2-(1, 1, 1-triphenyl-λ 5-phosphanylidene)-1 …
ZnCl2‐Promoted One‐Pot Three‐Component Synthesis of Multisubstituted Thiazolo[4,5‐b]pyridines and Thieno[2,3‐b:4,5‐b′]dipyridines
L Luo, L Meng, Y Peng, Y Xing, Q Sun… - European Journal of …, 2015 - Wiley Online Library
A ZnCl2‐promoted one‐pot synthesis of multisubstituted thiazolo [4, 5‐b] pyridines and
thieno [2, 3‐b: 4, 5‐b′] dipyridines from mercaptonitrile salts, α‐bromo ketones and ketones …
thieno [2, 3‐b: 4, 5‐b′] dipyridines from mercaptonitrile salts, α‐bromo ketones and ketones …
High Throughput Synthesis of Extended Pyrazolo[3,4-d]dihydropyrimidines
SV Ryabukhin, DS Granat, AS Plaskon… - ACS Combinatorial …, 2012 - ACS Publications
Thirteen 5-hetarylaminopyrazoles were synthesized in 62–93% yield through the arylation of
1-isopropyl-and 1-phenyl-5-aminopyrazoles with electrophilic hetarylhalides under …
1-isopropyl-and 1-phenyl-5-aminopyrazoles with electrophilic hetarylhalides under …
Synthesis of spiro[pyrazolo[3,4-b] pyridine-4,3′-indoline] and spiro [benzo[h]pyrazolo[3,4-b]quinoline-4,3′-indoline] derivatives using wet cyanuric chloride under …
Z Yin, L Yang, L Wu - Journal of Chemical Sciences, 2013 - Springer
A simple and efficient synthesis of spiro [pyrazolo [3, 4-b] pyridine-4, 3′-indoline] and spiro
[benzo [h] pyrazolo [3, 4-b] quinoline-4, 3′-indoline] derivatives has been accomplished by …
[benzo [h] pyrazolo [3, 4-b] quinoline-4, 3′-indoline] derivatives has been accomplished by …
Rapid synthesis of tetrahydroquinolines by indium trichloride catalyzed mono-and bis-intramolecular imino Diels–Alder reactions
RDRS Manian, J Jayashankaran, R Ramesh… - Tetrahedron letters, 2006 - Elsevier
A rapid synthesis of mono-and bis-tetrahydropyrazolo [4′, 3′: 5, 6] thiopyrano [4, 3-b]
quinolines has been achieved by the reaction of aldimines derived from aromatic amines …
quinolines has been achieved by the reaction of aldimines derived from aromatic amines …
3-Formylpyrazolo[1,5-a]pyrimidines as Key Intermediates for the Preparation of Functional Fluorophores
A one-pot route for the regioselective synthesis of 3-formylpyrazolo [1, 5-a] pyrimidines 4a–k
in good yields through a microwave-assisted process is provided. The synthesis proceeds …
in good yields through a microwave-assisted process is provided. The synthesis proceeds …
[引用][C] New one‐step synthesis of pyrazolo[1,5‐a]pyrimidine and pyrazolo[1,5‐a]quinazoline derivatives via multicomponent reactions
BK Ghotekar, MN Jachak… - Journal of Heterocyclic …, 2009 - Wiley Online Library
A series of pyrazolopyrimidine and pyrazoloquinozoline derivatives has been synthesized in
one step by multicomponent reactions using, 5‐aminopyrazole, p …
one step by multicomponent reactions using, 5‐aminopyrazole, p …
A facile environment-friendly one-pot two-step regioselective synthetic strategy for 3,7-diarylpyrazolo[1,5-a]pyrimidines related to zaleplon and 3,6-diarylpyrazolo[1,5-a] …
AS Devi, S Kaping, JN Vishwakarma - Molecular diversity, 2015 - Springer
Aminopyrazoles required for the synthesis of pyrazolo 1, 5-a pyrimidines were obtained by
the reaction of enaminonitriles with hydrazine hydrate. The resulting aminopyrazoles are …
the reaction of enaminonitriles with hydrazine hydrate. The resulting aminopyrazoles are …
Recent synthetic methodologies for pyrazolo[1,5-a]pyrimidine
The development of new synthetic routes towards pyrazolo [1, 5-a] pyrimidines for their
biological and medicinal exploration is an attractive area for researchers. This review …
biological and medicinal exploration is an attractive area for researchers. This review …