In this study, a series of twenty-two ring-substituted 8-hydroxyquinoline-2-carboxanilides
was prepared and characterized. Primary in vitro screening of the synthesized compounds …

In this study, a series of twenty-two ring-substituted 6-hydroxynaphthalene-2-carboxanilides
was prepared and characterized. Primary in vitro screening of the synthesized compounds …

The article describes the design, synthesis, and characterization of a new series of 8‐
trifluoromethylquinoline substituted pyrazole‐3‐carboxamides (9a, 9b, 9c, 9d, 9e, 9f, 9g, 9h …

Additional structural modifications of the new chemical entity, 2, 8-dicyclopentyl-4-
methylquinoline (DCMQ; MIC= 6.25 μg/mL, M. tuberculosis H37Rv) resulted in the synthesis …

A number of 4-amino substituted 2, 8-bis (trifluoromethyl) quinoline derivatives were
synthesized and evaluated for their in vitro antimycobacterial activity against Mycobacterium …

ABSTRACT A series of novel substituted N-(3-acetyl-2-oxoquinolin-1 (2H)-yl) benzamide
(AJQC1-AJQC12) have been synthesized upon refluxing 3-acetyl-1-amino-quinolin-2-one …

Twelve novel substituted 2‐chloroquinoline‐3‐carboxamide derivatives were prepared from
acetanilides using the Vilsmeier–Haack reaction, producing 2‐chloro‐3‐carbaldehyde …

As a continuation of our research and with the aim of obtaining new anti-tuberculosis agents
which can improve the current chemotherapeutic anti-tuberculosis treatments, forty-three …

As a continuation of our research and with the aim of obtaining new antituberculosis agents
which can improve the current chemotherapeutic antituberculosis treatments, new series of …

To develop new potential antimycobacterial drugs, a series of pyrazinamide derivatives was
designed, synthesized and tested for their ability to inhibit the growth of selected …