Two alternative routes have been developed for the synthesis of trichotomine dimethyl ester
2. Both routes involve the synthesis of keto lactam 3 by reaction of the chiral imine 4 …

Publisher Summary This chapter describes those alkaloids that contain two nuclei derived
from tryptophan, and is organized approximately along the lines of a progressing …

l-Carbethoxymethyl-2-(/3-carbethoxyethyl)-l, 2, 3, 4-tetrahydro-/3-carboline has been
converted into two different tetra-cyclic/3-ketoesters by employing two sets of reaction …

A short route to tetracyclic ring substructures of C-mavacurine, Strychnos, and akuammiline-
type alkaloids, based on the addition of methyl 1-, 2-, or 3-indoleacetate anions to Ñ …

ALTERNATIVE PARTIAL SYNTHESIS OF BISINDOLE ALKALOIDS G. MASSIOT, JM
NUZILLARD, B. RICHARD and L. LE MEN-QLIVIER Laboratoire de Page 1 Tehahedrm Letters …

Although 7-substituted 1-acetyl-2, 3-dihydroindoles are suitable building blocks for the
synthesis of biologically interesting indole alkaloids2 having a substituent at the 7-position …

Keyword (fr) PREPARATION ALCALOIDE LACTAME REACTION ELECTROPHILE
HETEROCYCLE AZOTE ANGULAIRE COMPOSE PENTACYCLIQUE EPOXYDE …

In a relatively short period of time several bis-indole alkaloids, especially those from
Catharunfhus roseus G. Don, have became highly valuable agents in chemotherapy. The …

l-[/3-[. ZVa-(Phenylsulfonyl) indol-3-yl] ethyl]-2-cyano-A3-piperidmes 21 and 26 have been
used to mimic the two-step reaction sequence 7-* 8 (Scheme I) in which a 5, 6 …

The transformation of tryptophol (1) into indoloquinolizidines (4)(Scheme I) represents the
backbone of a general method of indole alkaloid synthesis. 4 As part of an endeavor to …