An efficient synthesis of fully substituted pyrazolo [3, 4-b] pyridin-5-amines from α-azidochalcones

M Adib, F Peytam - Tetrahedron, 2018 - Elsevier
A facile, mild and efficient procedure for the synthesis of fully substituted pyrazolo [3, 4-b]
pyridin-5-amines is reported. A mixture of an α-azidochalcone, a 5-aminopyrazole and t …

One‐Pot and Convenient Conversion of 5‐Azidopyrazole‐4‐carboxaldehyde to Pyrazolo[3,4‐b]pyridines

A Zheng, W Zhang, J Pan - Synthetic communications, 2006 - Taylor & Francis
A one‐pot and convenient synthesis of multisubstituted pyrazolo [3, 4‐b] pyridines in
moderate to high yields has been achieved by a two‐step reaction: diazo‐transfer of 5‐azido …

An Efficient Protocol for the Synthesis of Pyrazolo [1, 5-c] quinazolines by a Staudinger–Aza-Wittig–Dehydroaromatization Sequence

M Xu, A Chen, Z Ren, J Qiu, M Zu, Y Zhang, J Wang… - Synlett, 2021 - thieme-connect.com
The one-pot synthesis of azide-substituted dihydropyrazoles in isopropanol was performed
by using chalcones, hydrazine hydrate, and an acyl chloride at 0℃. Subsequent Staudinger …

[HTML][HTML] Facile one-pot synthesis of the pyrazolo[1,5-a]pyrazine scaffold

OV Zaremba, NY Gorobets, SS Kovalenko… - Chemistry of …, 2013 - Springer
A series of novel pyrazolo [1, 5-a] pyrazine derivatives has been synthesized using a facile
one-pot three-step protocol starting from pyrazole-3-carboxylic acids. The process occurs via …

Facile synthesis of 1-substituted 4, 5-diaminopyrazoles and its application toward the synthesis of pyrazolo [3, 4-b] pyrazines

TC Chien, RA Smaldone, LB Townsend - Tetrahedron letters, 2004 - Elsevier
1-Substituted 5-aminopyrazole-4-carbonylazides were prepared from the appropriate 5-
aminopyrazole-4-carboxylates. The acyl azides undergo a Curtius rearrangement followed …

Three‐component synthesis of arene‐linked pyrazolo[1,5‐a]pyrimidines

AAM Ahmed, AEM Mekky… - Journal of Heterocyclic …, 2023 - Wiley Online Library
In this study, we aimed to establish an efficient method for synthesizing two new series of
arene‐linked pyrazolo [1, 5‐a] pyrimidines. This was achieved by reacting 1 H‐pyrazole‐3, 5 …

Facile, novel and efficient synthesis of new pyrazolo [3, 4-b] pyridine products from condensation of pyrazole-5-amine derivatives and activated carbonyl groups

A Ghaedi, GR Bardajee, A Mirshokrayi, M Mahdavi… - RSC …, 2015 - pubs.rsc.org
An efficient synthesis of novel ethyl-1, 3, 4-triphenyl-1H-pyrazolo [3, 4-b] pyridine-6-
carboxylate products has been achieved via condensation of pyrazole-5-amine derivatives …

New synthetic approach to pyrazolo[1,5‐a]pyrazine derivatives from 2,2‐dichlorovinylacetophenones

A Guirado, M Vera, B Martiz, F Ródenas… - Journal of …, 2023 - Wiley Online Library
New efficient synthetic methods in pyrazoline and pyrazolopyrazine chemistry have been
developed starting from 2, 2‐dichlorovinylacetophenones 1, which were sequentially …

[引用][C] An efficient synthesis of new class of pyrazolo[3,4‐b]pyridine‐6‐one derivatives by a novel cascade reaction

F Shi, J Zhang, S Tu, R Jia, Y Zhang… - Journal of …, 2007 - Wiley Online Library
A novel cascade reaction of 4‐arylidene‐2‐phenyl‐1, 3‐oxazol‐5 (4H)‐one with 3‐methyl‐1‐
phenyl‐1H‐pyrazol‐5‐amine was described and a number of new pyrazolo [3, 4‐b] pyridine …

A novel and convenient synthesis of thiazolo [3, 2-a] pyrimidin-7-ones and pyrido [1, 2-a] pyrimidin-2-ones using Vilsmeier reagent

YY Weng, LM Ying, QX Chen, WK Su - Chinese Chemical Letters, 2012 - Elsevier
A novel and convenient synthesis of thiazolo[3,2-a]pyrimidin-7-ones and pyrido[1,2-a]pyrimidin-2-ones
using Vilsmeier reagent - ScienceDirect Skip to main contentSkip to article Elsevier logo …