Synthesis and bioactivities of novel pyrazole oxime derivatives containing a 1, 2, 3-thiadiazole moiety

H Dai, S Ge, G Li, J Chen, Y Shi, L Ye, Y Ling - Bioorganic & Medicinal …, 2016 - Elsevier
A series of new pyrazole oxime compounds bearing a 1, 2, 3-thiadiazole ring were
designed, synthesized, and evaluated for their insecticidal, acaricidal and antitumor …

Hantzsch and Schiff's reaction: synthesis, in vitro cytotoxic and antimicrobial activity of [1, 3, 4] oxadiazoline and [1, 3] thiazole derivatives

N Chidananda, B Poojary, V Sumangala… - Medicinal Chemistry …, 2014 - Springer
Two new series of compounds namely, 1-chloro-4-(3, 4-dichlorophenyl)-3, 4-
dihydronaphthalene incorporated [1, 3, 4] oxadiazoline 4a–j and [1, 3] thiazole 6a–j …

Synthesis and biological activity profile of novel triazole/quinoline hybrids

H Jamshidi, MR Naimi‐Jamal, M Safavi… - Chemical Biology & …, 2022 - Wiley Online Library
Based on the significant and diverse pharmacophore features of triazole ring and
considering the potent antimicrobial properties of quinoline scaffold, a novel series of 1, 2, 3 …

An efficient synthesis of 2, 4′-bi-1, 3-oxa (thia) zoles as scaffolds for bioactive products

S Peña, L Scarone, E Manta, G Serra - Chemistry of Heterocyclic …, 2011 - Springer
A rapid and efficient methodology to prepare 2, 4′-bi-1, 3-azoles as scaffolds for
biologically active marine natural products is described. Hantzsch reaction and oxidative …

8-Hydroxyquinoline 1, 2, 3-triazole derivatives with promising and selective antifungal activity

NM da Silva, CB Gentz, P Reginatto… - Medical …, 2021 - academic.oup.com
Fungal infections that affect humans and plants have increased significantly in recent
decades. However, these pathogens are still neglected when compared to other infectious …

[HTML][HTML] Synthesis and anticancer evaluation of new 1, 3, 4-oxadiazole derivatives

CE Stecoza, GM Nitulescu, C Draghici, MT Caproiu… - Pharmaceuticals, 2021 - mdpi.com
In order to develop novel chemotherapeutic agents with potent anticancer activities, a series
of new 2, 5-diaryl/heteroaryl-1, 3, 4-oxadiazoles were designed and synthesized. The …

Design and discovery of novel antifungal quinoline derivatives with acylhydrazide as a promising pharmacophore

YD Yang, YH He, KY Ma, H Li, ZJ Zhang… - Journal of Agricultural …, 2021 - ACS Publications
Inspired by natural 2-quinolinecarboxylic acid derivatives, a series of quinoline compounds
containing acylhydrazine, acylhydrazone, sulfonylhydrazine, oxadiazole, thiadiazole, or …

Novel amide derivatives containing 1, 3, 4-thiadiazole moiety: Design, synthesis, nematocidal and antibacterial activities

J Chen, C Yi, S Wang, S Wu, S Li, D Hu… - Bioorganic & Medicinal …, 2019 - Elsevier
A series of novel amide derivatives containing 1, 3, 4-thiadiazole moiety were synthesized
and their bioactivities were evaluated. The compound 34 exhibited good nematocidal …

A review on novel synthesis approaches and biological activities of 1, 2, 4-oxadiazole and 1, 3, 4-oxadiazole tailored compounds

T Chaudhary, PK Upadhyay - Current Organic Synthesis, 2022 - ingentaconnect.com
Rational design and synthesis of novel compounds with both effectivity and safety properties
have always been a formidable task in the development of drugs. Oxadiazoles are …

[引用][C] Synthesis and Biological Activities of Novel Pyrazole Oximes Containing Substituted Oxadiazole Moiety

H Dai, Y Ding, X Du, W Yao… - CHINESE …, 2018 - SCIENCE PRESS 16 …