Synthesis and anticandidal activity of new triazolothiadiazine derivatives
New triazolothiadiazine derivatives were synthesized via the ring closure reaction of 4-
amino-5-substituted-2, 4-dihydro-3H-1, 2, 4-triazol-3-thiones with phenacyl bromides. The …
amino-5-substituted-2, 4-dihydro-3H-1, 2, 4-triazol-3-thiones with phenacyl bromides. The …
Synthesis of New [1,2,4]Triazolo[3,4‐b][1,3,4]thiadiazines and Study of Their Anti‐Candidal and Cytotoxic Activities
New triazolothiadiazine derivatives 5a–h were synthesized from 4‐amino‐3‐(4‐pyridyl)‐5‐
mercapto‐4H‐1, 2, 4‐triazole (3) with substituted aryl hydrazonoyl chlorides 4a–h. The …
mercapto‐4H‐1, 2, 4‐triazole (3) with substituted aryl hydrazonoyl chlorides 4a–h. The …
Synthesis and evaluation of thiazole–pyrimidine derivatives as new anticandidal and cytotoxic agents
The aim of this study was to describe the synthesis of four new 2-(3, 4-diphenyl-3 H-thiazol-2-
ylidene) amino-4, 6-dimethylpyrimidine derivatives, which were screened for their …
ylidene) amino-4, 6-dimethylpyrimidine derivatives, which were screened for their …
Novel triazolothiadiazole and triazolothiadiazine derivatives containing pyridine moiety: design, synthesis, bactericidal and fungicidal activities
RM Abdelhameed, HA El-Sayed… - Current Bioactive …, 2018 - ingentaconnect.com
Background: One of the important chemical agents in designing of anti-convulsant,
antiatherosclerotic and anti-cancer drugs are pyridine derivatives. Alkyl and aryl derivatives …
antiatherosclerotic and anti-cancer drugs are pyridine derivatives. Alkyl and aryl derivatives …
α,α-Dibromoacetophenones mediated synthesis of some new 7H-7-alkoxy-3-alkyl/phenyl-6-aryl-s-triazolo[3,4-b][1,3,4]thiadiazines and their antimicrobial evaluation
R Pundeer, V Kiran, R Prakash, Sushma… - Medicinal Chemistry …, 2012 - Springer
A series of new 7 H-7-alkoxy-3-alkyl/phenyl-6-aryl-s-triazolo [3, 4-b][1, 3, 4] thiadiazines (3,
4) were synthesized by the reaction of various α, α-dibromoacetophenones 1 with 3 …
4) were synthesized by the reaction of various α, α-dibromoacetophenones 1 with 3 …
Synthesis and antifungal activity of some s-mercaptotriazolobenzothiazolyl amino acid derivatives
A Aboelmagd, IAI Ali, EMS Salem… - European Journal of …, 2013 - Elsevier
A series of s-triazolobenzothiazolylthioacetyl/propionyl amino acid derivatives were
synthesized with the aim of evaluating their antifungal activity. Their chemical structures …
synthesized with the aim of evaluating their antifungal activity. Their chemical structures …
Synthesis of new 2-thio-[1, 2, 4] triazolo [1, 5-c] quinazoline derivatives and its antimicrobial activity
L Antipenko, A Karpenko, S Kovalenko… - Chemical and …, 2009 - jstage.jst.go.jp
A series of novel ([1, 2, 4] triazolo [1, 5-c] quinazolin-2-ylthio) carboxylic acids 2a—d and
esters 3a—l were synthesized and evaluated for antimicrobial activity. Alkylation of …
esters 3a—l were synthesized and evaluated for antimicrobial activity. Alkylation of …
Synthesis and biological evaluation of a new series of pyrazolines as new anticandidal agents
New pyrazoline derivatives bearing an oxadiazole moiety were synthesized via the reaction
of 1-(chloroacetyl)-3-(2-furyl/thienyl)-5-aryl-2-pyrazolines with 5-substituted-1, 3, 4 …
of 1-(chloroacetyl)-3-(2-furyl/thienyl)-5-aryl-2-pyrazolines with 5-substituted-1, 3, 4 …
[PDF][PDF] Synthesis of Some Novel Bis [1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazine Derivatives for Antimicrobial Evaluation
CS Reddy, DC Rao, V Yakub… - Acta Chimica …, 2011 - acta-arhiv.chem-soc.si
A new series of novel bis [1, 2, 4] triazolo [3, 4-b][1, 3, 4] thiadiazines 7a–j has been
synthesized by the reaction of [5, 5'-methylenebis (3-methylbenzofuran-7, 5-diyl)] bis [(4 …
synthesized by the reaction of [5, 5'-methylenebis (3-methylbenzofuran-7, 5-diyl)] bis [(4 …
Synthesis and antimicrobial activity of 4-phenyl/cyclohexyl-5-(1-phenoxyethyl)-3-[N-(2-thiazolyl) acetamido] thio-4H-1, 2, 4-triazole derivatives
The increasing clinical importance of drug-resistant fungal and bacterial pathogens has lent
additional urgency to microbiological research and new antimicrobial compound …
additional urgency to microbiological research and new antimicrobial compound …