Synthesis, molecular docking and antimicrobial evaluation of novel benzoxazole derivatives
T Ertan-Bolelli, I Yildiz, S Ozgen-Ozgacar - Medicinal Chemistry Research, 2016 - Springer
In this research, previously and newly synthesized 5-amino-2-(4-substitutedphenyl/benzyl)
benzoxazoles (3a–3l) and 2-substituted-5-(4-nitro/aminophenylsulfonamido) benzoxazoles …
benzoxazoles (3a–3l) and 2-substituted-5-(4-nitro/aminophenylsulfonamido) benzoxazoles …
Design, synthesis and mode of action of some benzothiazole derivatives bearing an amide moiety as antibacterial agents
In this study ten benzothiazole derivatives bearing the amide moiety were designed,
synthesized and evaluated for their antibacterial activity and possible mode of action …
synthesized and evaluated for their antibacterial activity and possible mode of action …
Synthesis and antimicrobial evaluation of novel 5-substituted-2-(p-tert-butylphenyl)benzoxazoles
M Taşcı, O Temiz-Arpaci, F Kaynak-Onurdag, S Okten - 2018 - nopr.niscpr.res.in
In the present study, a series of nine novel 5-substituted-2-(p-tert-butylphenyl) benzoxazole
derivatives have been synthesized and their structures confirmed by spectral techniques …
derivatives have been synthesized and their structures confirmed by spectral techniques …
[PDF][PDF] Synthesis, characterization and anti-microbial activity of novel substituted benzoxazole derivatives
G Balaswamy, K Srinivas, P Pradeep… - International Journal of …, 2012 - hakon-art.com
In view of the fact that a large number of derivatives of benzoxazole have been found to
exhibit a wide variety of pharmacological activities. In the current research work, the title …
exhibit a wide variety of pharmacological activities. In the current research work, the title …
Synthesis, molecular docking, and DFT studies of some new 2, 5-disubstituted benzoxazoles as potential antimicrobial and cytotoxic agents
In this study, a total of 17 piece 2, 5-disubstituted benzoxazole derivatives were synthesized,
2 of which were not original, their antimicrobial activities were determined using …
2 of which were not original, their antimicrobial activities were determined using …
Synthesis and antimicrobial activity of some novel 2, 5-and/or 6-substituted benzoxazole and benzimidazole derivatives
A new series of 2, 5-and/or 6-substituted benzoxazoles (7a–f), benzimidazoles (8a–g)
holding cyclohexyl or cyclopentyl moieties at position 2 and 5-or 6-substituted-2 …
holding cyclohexyl or cyclopentyl moieties at position 2 and 5-or 6-substituted-2 …
New vinyl-1, 2, 4-triazole derivatives as antimicrobial agents: Synthesis, biological evaluation and molecular docking studies
E Stingaci, M Zveaghinteva, S Pogrebnoi… - Bioorganic & Medicinal …, 2020 - Elsevier
Triazole is a very important scaffold in medicinal chemistry due to the wide spectrum of
biological activities and mainly antifungal activity of 1, 2, 4-triazole derivatives. The main …
biological activities and mainly antifungal activity of 1, 2, 4-triazole derivatives. The main …
Design, synthesis and biological potential of heterocyclic benzoxazole scaffolds as promising antimicrobial and anticancer agents
Background Benzoxazole is the most important class of heterocyclic compound in medicinal
chemistry. It has been incorporated in many medicinal compounds making it a versatile …
chemistry. It has been incorporated in many medicinal compounds making it a versatile …
Design and Synthesis of Benzoxepine–Based 1, 2, 3‐Triazoles: Molecular Docking and in vitro Antimicrobial Activity Evaluation
SK Gandham, AA Kudale, T Rao Allaka… - ChemistrySelect, 2022 - Wiley Online Library
Here, we report a novel series of dihydrobenzoxepin linked to 1, 2, 3‐triazole scaffolds (5 a‐
k) along with their pharmacological activity against different Gram–(+ ve), Gram–(–ve) and …
k) along with their pharmacological activity against different Gram–(+ ve), Gram–(–ve) and …
Synthesis of new benzimidazole derivatives containing 1, 3, 4-thiadiazole: their in vitro antimicrobial, in silico molecular docking and molecular dynamic simulations …
ABSTRACT A series of some new benzimidazole-1, 3, 4-thiadiazoles was synthesized. The
structures of target substances were confirmed by using 1H-NMR and 13С-NMR …
structures of target substances were confirmed by using 1H-NMR and 13С-NMR …