Synthesis, molecular docking and antimicrobial evaluation of novel benzoxazole derivatives

T Ertan-Bolelli, I Yildiz, S Ozgen-Ozgacar - Medicinal Chemistry Research, 2016 - Springer
In this research, previously and newly synthesized 5-amino-2-(4-substitutedphenyl/benzyl)
benzoxazoles (3a–3l) and 2-substituted-5-(4-nitro/aminophenylsulfonamido) benzoxazoles …

Design, synthesis and mode of action of some benzothiazole derivatives bearing an amide moiety as antibacterial agents

M Singh, SK Singh, M Gangwar, G Nath, SK Singh - RSC advances, 2014 - pubs.rsc.org
In this study ten benzothiazole derivatives bearing the amide moiety were designed,
synthesized and evaluated for their antibacterial activity and possible mode of action …

Synthesis and antimicrobial evaluation of novel 5-substituted-2-(p-tert-butylphenyl)benzoxazoles

M Taşcı, O Temiz-Arpaci, F Kaynak-Onurdag, S Okten - 2018 - nopr.niscpr.res.in
In the present study, a series of nine novel 5-substituted-2-(p-tert-butylphenyl) benzoxazole
derivatives have been synthesized and their structures confirmed by spectral techniques …

[PDF][PDF] Synthesis, characterization and anti-microbial activity of novel substituted benzoxazole derivatives

G Balaswamy, K Srinivas, P Pradeep… - International Journal of …, 2012 - hakon-art.com
In view of the fact that a large number of derivatives of benzoxazole have been found to
exhibit a wide variety of pharmacological activities. In the current research work, the title …

Synthesis, molecular docking, and DFT studies of some new 2, 5-disubstituted benzoxazoles as potential antimicrobial and cytotoxic agents

M Erol, I Celik, E Uzunhisarcikli… - Polycyclic Aromatic …, 2022 - Taylor & Francis
In this study, a total of 17 piece 2, 5-disubstituted benzoxazole derivatives were synthesized,
2 of which were not original, their antimicrobial activities were determined using …

Synthesis and antimicrobial activity of some novel 2, 5-and/or 6-substituted benzoxazole and benzimidazole derivatives

İ Ören, Ö Temiz, I Yalçın, E Şener, N Altanlar - European journal of …, 1999 - Elsevier
A new series of 2, 5-and/or 6-substituted benzoxazoles (7a–f), benzimidazoles (8a–g)
holding cyclohexyl or cyclopentyl moieties at position 2 and 5-or 6-substituted-2 …

New vinyl-1, 2, 4-triazole derivatives as antimicrobial agents: Synthesis, biological evaluation and molecular docking studies

E Stingaci, M Zveaghinteva, S Pogrebnoi… - Bioorganic & Medicinal …, 2020 - Elsevier
Triazole is a very important scaffold in medicinal chemistry due to the wide spectrum of
biological activities and mainly antifungal activity of 1, 2, 4-triazole derivatives. The main …

Design, synthesis and biological potential of heterocyclic benzoxazole scaffolds as promising antimicrobial and anticancer agents

S Kakkar, S Kumar, B Narasimhan, SM Lim… - Chemistry Central …, 2018 - Springer
Background Benzoxazole is the most important class of heterocyclic compound in medicinal
chemistry. It has been incorporated in many medicinal compounds making it a versatile …

Design and Synthesis of Benzoxepine–Based 1, 2, 3‐Triazoles: Molecular Docking and in vitro Antimicrobial Activity Evaluation

SK Gandham, AA Kudale, T Rao Allaka… - ChemistrySelect, 2022 - Wiley Online Library
Here, we report a novel series of dihydrobenzoxepin linked to 1, 2, 3‐triazole scaffolds (5 a‐
k) along with their pharmacological activity against different Gram–(+ ve), Gram–(–ve) and …

Synthesis of new benzimidazole derivatives containing 1, 3, 4-thiadiazole: their in vitro antimicrobial, in silico molecular docking and molecular dynamic simulations …

U Acar Çevik, A Işık, AE Evren, Ö Kapusız… - SAR and QSAR in …, 2022 - Taylor & Francis
ABSTRACT A series of some new benzimidazole-1, 3, 4-thiadiazoles was synthesized. The
structures of target substances were confirmed by using 1H-NMR and 13С-NMR …