Functional characterization of the A2b adenosine receptor in NIH 3T3 fibroblasts

LE Brackett, JW Daly - Biochemical pharmacology, 1994 - Elsevier
The adenosine (ADO) receptor in NIH 3T3 fibroblasts was characterized using a series of
adenosine agonists and selected xanthine and non-xanthine antagonists. The ADO receptor …

Functional characterization of adenosine A2 receptors in Jurkat cells and PC12 cells using adenosine receptor agonists

I van der Ploeg, S Ahlberg, FE Parkinson… - Naunyn-Schmiedeberg's …, 1996 - Springer
The effect of several adenosine analogues on cyclic AMP accumulation was examined in
the rat phaeochromocytoma cell PC12 and in the human T-cell leukaemia cell Jurkat …

[PDF][PDF] Potent adenosine receptor antagonists that are selective for the A1 receptor subtype.

EA Martinson, RA Johnson, JN Wells - Molecular pharmacology, 1987 - Citeseer
The xanthines currently represent the most potent class of adenosine receptor antagonists.
However, known derivatives of xanthine show little difference in antagonist potency between …

[HTML][HTML] A2A adenosine receptors from rat striatum and rat pheochromocytoma PC12 cells: characterization with radioligand binding and by activation of adenylate …

I HIDE, WL PADGETI, KA JACOBSON… - Molecular …, 1992 - ncbi.nlm.nih.gov
A2A Adenosine Receptors from Rat Striatum and Rat Pheochromocytoma PC12 Cells:
Characterization with Radioligand Binding and by Activation of Adenylate Cyclase - PMC Back …

Cloning and expression of an A1 adenosine receptor from rat brain.

LC Mahan, LD McVittie, EM Smyk-Randall… - Molecular …, 1991 - ASPET
We have used the polymerase chain reaction technique to selectively amplify guanine
nucleotide-binding regulatory protein (G protein)-coupled receptor cDNA sequences from rat …

Characterization of the A2B adenosine receptor from mouse, rabbit, and dog

JA Auchampach, LM Kreckler, TC Wan, JE Maas… - … of Pharmacology and …, 2009 - ASPET
We have cloned and pharmacologically characterized the A2B adenosine receptor (AR)
from the dog, rabbit, and mouse. The full coding regions of the dog and mouse A2BAR were …

[HTML][HTML] The A1 adenosine receptor. Solubilization and characterization of a guanine nucleotide-sensitive form of the receptor.

GL Stiles - Journal of Biological Chemistry, 1985 - Elsevier
Adenosine acting through membrane-bound A1 receptors is capable of inhibiting the
enzyme adenylate cyclase. A1 adenosine receptors from rat cerebral cortex have been …

[HTML][HTML] Demonstration of both A1 and A2 adenosine receptors in DDT1 MF-2 smooth muscle cells

V Ramkumar, WW Barrington, KA Jacobson… - Molecular …, 1990 - ncbi.nlm.nih.gov
Adenosine receptors of the A 1, and A 2 subtypes were characterized in membranes from
DDT 1, MF-2 smooth muscle cells. These cells possess a high density of A 1, adenosine …

A selective agonist affinity label for A3 adenosine receptors

XD Ji, C Gallorodriguez, KA Jacobson - Biochemical and biophysical …, 1994 - Elsevier
A newly synthesized, chemically reactive adenosine derivative, N 6-(3-
isothiocyanatobenzyl) adenosine-5′-N-methyluronamide, was found to bind selectively to …

Potent antagonists for the human adenosine A2B receptor. Derivatives of the triazolotriazine adenosine receptor antagonist ZM241385 with high affinity

M De Zwart, RC Vollinga, MW Beukers… - Drug development …, 1999 - Wiley Online Library
A series of novel and known 5‐substituted 7‐amino‐2‐(2‐furyl)[1, 2, 4] triazolo [1, 5‐a][1, 3,
5] triazine derivatives were synthesized and tested for adenosine receptor antagonism in …