Building on our previous work that discovered 1, 2, 4-triazole–spirodienone as a promising
pharmacophore for anticancer activity, we have further diversified 1, 2, 4–triazole …

In this article, we continued our previous effort to develop new selective anticancer
candidates based on the basic pharmacophoric requirements of both EGFR and VEGFR-2 …

In the current study, new benzimidazole-based 1, 3, 4-oxadiazole derivatives have been
synthesized and characterized by NMR, IR, MS, and elemental analysis. The final …

Two series of novel tricyclic oxazine and oxazepine fused quinazolines have been designed
and synthesized. The in vitro antitumor effect of the title compounds was screened on N87 …

A novel group of indolyl‐1, 2, 4‐triazole‐chalcone hybrids was designed, synthesized, and
assessed for their anticancer activity. The synthesized compounds exhibited significant …

A series of 1H-1, 2, 3-triazole-4H-chromene-D-glucose hybrid compounds 7a-o was
synthesized via click chemistry using 2-amino-7-propargyloxy-4H-chromene-3-carbonitriles …

A general strategy was developed for the synthesis of new fully decorated 1, 2, 3-triazoles
(5a-m & 6a-e) containing coumarine and sulfonyl-benzimidazole from 3-(2-((1-methyl-1H …

New quinoline/chalcone hybrids containing 1, 2, 4-triazole moiety have been designed,
synthesized and their structures elucidated and confirmed by various spectroscopic …

New series of isoxazole derivatives were synthesized and evaluated for in vitro antitumor
activity against HepG2, MCF-7 and HCT-116 cancer cells. Results showed that 4b and 25a …

This study represents the synthetic approaches of a new set of 2-(((3-(benzofuran-2-yl)-1-
phenyl-1H-pyrazol-4-yl) methylene) hydrazono)-5-(aryl) thiazolidin-4-one derivatives 4–22 …