New hydrazide–hydrazones of isonicotinic acid: Synthesis, lipophilicity and in vitro antimicrobial screening

Ł Popiołek, A Biernasiuk, A Berecka… - Chemical Biology & …, 2018 - Wiley Online Library
This study describes the synthesis, lipophilicity and in vitro antimicrobial assays of 15 new
hydrazide–hydrazones of isonicotinic acid. New derivatives were obtained on the basis of …

Synthesis, antimycobacterial activity and docking study of 2-aroyl-[1] benzopyrano [4, 3-c] pyrazol-4 (1H)-one derivatives and related hydrazide-hydrazones

VT Angelova, V Valcheva, T Pencheva… - Bioorganic & Medicinal …, 2017 - Elsevier
A new convenient method for preparation of 2-aroyl-[1] benzopyrano [4, 3-c] pyrazol-4 (1H)-
one derivatives 5b–g and coumarin containing hydrazide-hydrazone analogues 4a–e was …

Synthesis, antimycobacterial, antiviral, antimicrobial activities, and QSAR studies of isonicotinic acid-1-(substituted phenyl)-ethylidene/cycloheptylidene hydrazides

V Judge, B Narasimhan, M Ahuja, D Sriram… - Medicinal Chemistry …, 2012 - Springer
A series of isonicotinic acid-1-(substituted phenyl)-ethylidene/cycloheptylidene hydrazide
derivatives (1–12) was tested for their, in vitro antimycobacterial activity against …

Novel 4-(morpholin-4-yl)-N′-(arylidene) benzohydrazides: synthesis, antimycobacterial activity and QSAR investigations

V Raparti, T Chitre, K Bothara, V Kumar… - European journal of …, 2009 - Elsevier
A series of 4-(morpholin-4-yl)-N′-(arylidene) benzohydrazides were synthesized using
appropriate synthetic route. Antimycobacterial activity of the synthesized compounds (5a–5j) …

[引用][C] Synthesis and antitubercular activity of isonicotinoyl and cyanoacetyl hydrazones

D Chakravarty, A Bose, S Bose - Journal of pharmaceutical sciences, 1964 - Elsevier
Synthesis and Antitubercular Activity of Isonicotinoyl and Cyanoacetyl Hydrazones Page 1
1036 Journal of Pharmaceutical Skes Examination of the Oil.-The red basil oil which Ocimum …

Synthesis and antimycobacterial activities of some new thiazolylhydrazone derivatives

K Ozadali, OU Tan, P Yogeeswari… - Bioorganic & medicinal …, 2014 - Elsevier
This Letter reports the synthesis and evaluation of some thiazolylhydrazone derivatives for
their in vitro antimycobacterial activities against Mycobacterium tuberculosis H37Rv. The …

N-Substituted 2-Isonicotinoylhydrazinecarboxamides — New Antimycobacterial Active Molecules

Z Rychtarčíková, M Krátký, M Gazvoda, M Komlóová… - Molecules, 2014 - mdpi.com
This report presents a new modification of the isoniazid (INH) structure linked with different
anilines via a carbonyl group obtained by two synthetic procedures and with N-substituted 5 …

Synthesis and antimycobacterial activity of some coupling products from 4-aminobenzoic acid hydrazones

ŞG Küçükgüzel, S Rollas, I Küçükgüzel… - European journal of …, 1999 - Elsevier
Various 2, 3, 4-pentanetrione-3-[4-[[(5-nitro-2-furyl/pyridyl/substituted phenyl) methylene]
hydrazinocarbonyl] phenyl] hydrazones 3a–j were synthesized by the reactions of …

Synthesis and characterization of novel hydrazone derivatives of isonicotinic hydrazide and their evaluation for antibacterial and cytotoxic potential

MA Shah, A Uddin, MR Shah, I Ali, R Ullah, PA Hannan… - Molecules, 2022 - mdpi.com
Hydrazones are active compounds having an azomethine–NHN= CH group and are widely
studied owing to their ease of preparation and diverse pharmacological benefits. Novel …

Synthesis and antituberculosis activity of new hydrazide derivatives

ZA Kaplancikli, G Turan‐Zitouni… - … der Pharmazie: An …, 2008 - Wiley Online Library
The increasing clinical importance of drug‐resistant mycobacterial pathogens, especially
Mycobacterium tuberculosis, has lent additional urgency to microbiological research and …