Abstract LBT‐999 (8‐((E)‐4‐fluoro‐but‐2‐enyl)‐3β‐p‐tolyl‐8‐aza‐bicyclo [3.2. 1] octane‐2β‐
carboxylic acid methyl ester) is a cocaine derivative belonging to a new generation of highly …

Abstract LBT‐999 (8‐((E)‐4‐fluoro‐but‐2‐enyl)‐3‐beta‐p‐tolyl‐8‐aza‐bicyclo [3.2. 1]
octane‐2‐beta‐carboxylicacid methyl ester) is a recently developed cocaine derivative …

LBT-999 (8-((E)-4-fluoro-but-2-enyl)-3β-p-tolyl-8-aza-bicyclo [3.2. 1] octane-2β-carboxylic
acid methyl ester), a cocaine derivative belonging to a new generation of highly selective …

BACKGROUND: LBT-999 (E)-N-(4-fluorobut-2-enyl)-2β-carbomethoxy-3β-(4′-tolyl)
nortropane is a dopamine transporter (DAT) ligand.[18F] LBT-999 was first labelled with …

In this study the N‐fluoropropyl analogue of the cocaine congener β‐CFT (I), N‐(3‐
fluoropropyl)‐2β‐carbomethoxy‐3β‐(4‐fluorophenyl) nortropane (β‐CFT‐FP, III), was …

INTRODUCTION: LBT-999,(E)-N-(4-fluorobut-2-enyl)-2β-carbomethoxy-3β-(4'-tolyl)
nortropane, has been developed for PET imaging of the dopamine transporter.[18F] LBT …

The synthesis and 11C‐radiolabelling of a new tropane analogue, 3β‐(4′‐chlorophenyl)‐
2β‐(3′‐phenylisoxazol‐5′‐yl) tropane)(β‐CPPIT), an inhibitor of the dopamine …

Abstract PE2I ((E)‐N‐(3‐iodoprop‐2‐enyl)‐2β‐(4′‐tolyl) nortropane) is a cocaine
derivative belonging to a new generation of selective dopamine transporter inhibitors …

The compound 3β-(4′-chlorophenyl)-2β-(3′-phenylisoxazol-5′-yl) tropane (CPPIT or RTI
177) is a 2β-heterocyclic substituted cocaine congener with high in vitro selectivity and …

The fluoroalkyl-containing tropane derivative 2β-carbo-2′-fluoroethoxy-3β-(4-bromo-
phenyl) tropane (MCL-322) is a highly potent and moderately selective ligand for the …