Neurokinin B‐ and specific tachykinin NK3 receptor agonists‐induced airway hyperresponsiveness in the guinea‐pig
S Daoui, E Naline, V Lagente… - British journal of …, 2000 - Wiley Online Library
… Tachykinins induce … NK 3 receptor agonists to induce the development of airway
hyperresponsiveness. In the present study, we found that NKB and the tachykinin NK 3 receptor …
hyperresponsiveness. In the present study, we found that NKB and the tachykinin NK 3 receptor …
Potency and selectivity of the tachykinin NK3 receptor antagonist SR 142801
JC Beaujouan, M Saffroy, Y Torrens… - European journal of …, 1997 - Elsevier
… Other authors have indicated that SR 48968 antagonizes the release of Ca 2+ from inositol
trisphosphate-sensitive intracellular stores evoked by tachykinin NK 3 receptor agonists in …
trisphosphate-sensitive intracellular stores evoked by tachykinin NK 3 receptor agonists in …
Molecular and pharmacological characterization of the murine tachykinin NK3 receptor
HM Sarau, JA Feild, RS Ames, JJ Foley… - European journal of …, 2001 - Elsevier
… NK 3 receptors, respectively. Binding affinities and functional potencies of tachykinin receptor
agonists … ) 293 cells expressing murine NK 3 receptor and human NK 3 receptor, although …
agonists … ) 293 cells expressing murine NK 3 receptor and human NK 3 receptor, although …
Cardiovascular and behavioural effects of intracerebroventricularly administered tachykinin NK3 receptor antagonists in the conscious rat
E Cellier, L Barbot, D Regoli… - British journal of …, 1997 - Wiley Online Library
… Antagonist activities of SR142801 have been shown in various functional NK 3 receptor
agonist-evoked responses, notably the contraction of the guinea-pig ileum and of the rat portal …
agonist-evoked responses, notably the contraction of the guinea-pig ileum and of the rat portal …
Tachykinin neurokinin 3 receptor antagonists: a patent review (2005–2010)
P Malherbe, TM Ballard, H Ratni - Expert Opinion on Therapeutic …, 2011 - Taylor & Francis
… used to derive novel NK 3 receptor antagonists which have … agonist with the highest affinity
for the NK 3 receptor, binding … selective and potent agonist at the NK 3 receptor with a pK i …
for the NK 3 receptor, binding … selective and potent agonist at the NK 3 receptor with a pK i …
Neurokinin-3 receptor antagonists
GAM Giardina, LF Raveglia - Expert Opinion on Therapeutic …, 1997 - Taylor & Francis
… NK3 receptor agonists, a number of potential therapeutic indications for NK3 receptor …
research explosion in the tachykinin area was mainly on NK1 and NK2 receptors, to a large …
research explosion in the tachykinin area was mainly on NK1 and NK2 receptors, to a large …
GR138676, a novel peptidic tachykinin antagonist which is potent at NK3 receptors
JM Stables, IJM Beresford, S Arkinstall, SJ Ireland… - Neuropeptides, 1994 - Elsevier
… of tachykinin agonists, including the NK3 receptorpreferring … tachykinin antagonist, GR138676,
antagonised NK, receptor-… reported that tachykinin agonists bound to NK, receptors in …
antagonised NK, receptor-… reported that tachykinin agonists bound to NK, receptors in …
The study of tachykinin receptors
E Burcher - Clinical and experimental pharmacology and …, 1989 - Wiley Online Library
… peripheral NK3 receptors have been described. In contrast, NKI, NK3 but not NK2 receptors
… A number of more selective peptide analogue agonists has been synthesised, for example, […
… A number of more selective peptide analogue agonists has been synthesised, for example, […
… tachykinin receptor antagonists: I. Pharmacological and pharmacokinetic characterization of SB 223412, a novel, potent and selective neurokinin-3 receptor …
HM Sarau, DE Griswold, W Potts, JJ Foley… - … of Pharmacology and …, 1997 - ASPET
… of behavioral responses induced by the NK-3 receptor-selective agonist, senktide (ED 50 =
… and pathophysiological roles of NK-3 receptors. The mammalian tachykinins, also known as …
… and pathophysiological roles of NK-3 receptors. The mammalian tachykinins, also known as …
SCH 206272: a potent, orally active tachykinin NK1, NK2, and NK3 receptor antagonist
JC Anthes, RW Chapman, C Richard, S Eckel… - European journal of …, 2002 - Elsevier
… at human tachykinin NK 1 , NK 2 , and NK 3 receptors (K i =… cloned human tachykinin NK 1
, NK 2 , or NK 3 receptors. SCH … ±0.3) induced by the tachykinin NK 1 receptor agonist, [Met-O-…
, NK 2 , or NK 3 receptors. SCH … ±0.3) induced by the tachykinin NK 1 receptor agonist, [Met-O-…
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