Effects of central administration of tachykinin receptor agonists and antagonists on plus-maze behavior in mice

RM Teixeira, ARS Santos, SJ Ribeiro, JB Calixto… - European journal of …, 1996 - Elsevier
… None of the tachykinin receptor agonists or antagonists modified … NK~ and NK 2 receptor
agonists and antagonists can modulate … Stimulation of either tachykinin NK 1 or NK 2 receptors

Tachykinin receptors antagonists: from research to clinic

L Quartara, M Altamura - Current drug targets, 2006 - ingentaconnect.com
tachykinin NK-2 receptor, with high selectivity vs. the tachykinin NK-1 and NK-3 receptors.
The compound was active in vivo in several animal models of NK-2 agonist induced effects [93…

Tachykinins and tachykinin receptors: structure and activity relationships

TA Almeida, J Rojo, PM Nieto, FM Pinto… - Current medicinal …, 2004 - ingentaconnect.com
… and that both tachykinins and their receptors are of peptide … on evolution of tachykinin and
tachykinin receptor sequences. … tachykinins is that they are able to act as full agonists, albeit …

The tachykinin NK1 receptor in the brain: pharmacology and putative functions

A Saria - European journal of pharmacology, 1999 - Elsevier
agonists served to further characterize tachykinin receptor … SP or selective tachykinin NK 1
receptor agonists. Locomotion… administration of tachykinin NK 1 receptor agonists, probably …

Tachykinin receptor antagonists in clinical trials

L Quartara, M Altamura, S Evangelista… - Expert opinion on …, 2009 - Taylor & Francis
… In vivo, ibodutant inhibited visceral muscle contractions induced by NK2 receptor agonists,
with high potency and long duration of action, after either iv or oral administration Citation[101]…

Molecular recognition of tachykinin receptor selective agonists: insights from structural studies

A Ganjiwale, SM Cowsik - Mini reviews in medicinal chemistry, 2013 - ingentaconnect.com
agonists important for receptor binding and biological activity is of great significance in
unraveling the molecular mechanisms involved in tachykinin receptor … and NK2 receptor agonists. …

Tachykinin receptors and the airways

N Frossard, C Advenier - Life sciences, 1991 - Elsevier
… 2 receptor agonists produce concentrationdependent contraction (80). NK-3 receptor agonists
… the natural tachykinins (83) and to the NK-2 selective agonist used (84). Inhibitory effect of …

Tachykinin receptors antagonism for asthma: a systematic review

R Ramalho, R Soares, N Couto, A Moreira - BMC pulmonary medicine, 2011 - Springer
… This review systematically examines randomized controlled trials evaluating the effect of
tachykinins receptors antagonism on asthma. Symptoms, airway inflammation, lung function …

Pharmacology of tachykinin receptors on neurones in the ventral tegmental area of rat brain slices

GR Seabrook, BJ Bowery, RG Hill - European journal of pharmacology, 1995 - Elsevier
tachykinin receptor agonists on dopamine neurones within the rat ventral tegmental area. …
tachykinin receptor agonists. However, a major complication with these studies is that agonists

The tachykinin peptide family, with particular emphasis on mammalian tachykinins and tachykinin receptor agonists

JM Conlon - Tachykinins, 2004 - Springer
agonists for the NK 2 receptor. The NH 2 terminal extension to the NKA sequence in these
tachykinins has only minor effects on potency in vitro but the greater stability of these agonists