Novel C-17-heteroaryl steroidal CYP17 inhibitors/antiandrogens: synthesis, in vitro biological activity, pharmacokinetics, and antitumor activity in the LAPC4 human …

VD Handratta, TS Vasaitis, VCO Njar… - Journal of medicinal …, 2005 - ACS Publications
New chemical entities, steroidal C-17 benzoazoles (5, 6, 9 and 10) and pyrazines (14 and
15) were rationally designed and synthesized. The key reaction for synthesis of the …

[引用][C] Novel C-17-heteroaryl steroidal CYP17 inhibitors/antiandrogens: Synthesis, in vitro biological activity, pharmacokinetics, and antitumor activity in the LAPC4 …

VD HANDRATTA, TS VASAITIS… - Journal of medicinal …, 2005 - pascal-francis.inist.fr
Novel C-17-heteroaryl steroidal CYP17 inhibitors/antiandrogens : Synthesis, in vitro
biological activity, pharmacokinetics, and antitumor activity in the LAPC4 human prostate …

[引用][C] Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens: Synthesis, in Vitro Biological Activity, Pharmacokinetics, and Antitumor Activity in the LAPC4 …

VD Handratta, TS Vasaitis, VCO Njar… - Journal of Medicinal …, 2005 - infona.pl
Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens: Synthesis, in Vitro Biological
Activity, Pharmacokinetics, and Antitumor Activity in the LAPC4 Human Prostate Cancer …

[引用][C] Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens: Synthesis, in Vitro Biological Activity, Pharmacokinetics, and Antitumor Activity in the LAPC4 …

VD Handratta, TS Vasaitis, VCO Njar… - Journal of Medicinal …, 2005 - cir.nii.ac.jp
Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens: Synthesis, in Vitro Biological
Activity, Pharmacokinetics, and Antitumor Activity in the LAPC4 Human Prostate Cancer …

Novel C-17-heteroaryl steroidal CYP17 inhibitors/antiandrogens: synthesis, in vitro biological activity, pharmacokinetics, and antitumor activity in the LAPC4 human …

VD Handratta, TS Vasaitis, VC Njar… - Journal of Medicinal …, 2005 - europepmc.org
New chemical entities, steroidal C-17 benzoazoles (5, 6, 9 and 10) and pyrazines (14 and
15) were rationally designed and synthesized. The key reaction for synthesis of the …

Novel C-17-heteroaryl steroidal CYP17 inhibitors/antiandrogens: synthesis, in vitro biological activity, pharmacokinetics, and antitumor activity in the LAPC4 human …

VD Handratta, TS Vasaitis, VCO Njar… - Journal of …, 2005 - pubmed.ncbi.nlm.nih.gov
New chemical entities, steroidal C-17 benzoazoles (5, 6, 9 and 10) and pyrazines (14 and
15) were rationally designed and synthesized. The key reaction for synthesis of the …

[引用][C] Novel C-17-heteroaryl steroidal CYP17 inhibitors/antiandrogens: Synthesis, in vitro biological activity, pharmacokinetics, and antitumor activity in the LAPC4 …

VD HANDRATTA, TS VASAITIS… - Journal of …, 2005 - American Chemical Society