Novel Sulfoximine Derivatives Containing Cyanoguanidine and Nitroguanidine Moieties: Design, Synthesis, and Bioactivities

Y Xie, H Li, D Liu, L Zhao, X Liu, X Liu… - Journal of Agricultural …, 2024 - ACS Publications
A total of 32 novel sulfoximines bearing cyanoguanidine and nitroguanidine moieties were
designed and synthesized by a rational molecule design strategy. The bioactivities of the …

Design, synthesis, and antifungal activities of novel sulfoximine derivatives for plant protection

Y Liu, H Li, Y Zhao, Y Xie, Y He, Y Qin… - Pest Management …, 2023 - Wiley Online Library
BACKGROUND Fungicides play a significant role in the integrated management of plant
pathogens. However, the irrational application of fungicides with similar structures has led to …

Design, synthesis, and antifungal activity of sulfoximine derivatives containing nitroguanidine moieties

Y Xiao, H Li, Q Shao, Y Liu, Y Xie… - Chemistry & …, 2022 - Wiley Online Library
To discover novel pesticide candidates, a series of sulfoximine derivatives were designed
and synthesized via the oxidation coupling reaction of sulfides and N‐alkyl nitroguanidines …

Design, synthesis, and biological activity of sulfoximine derivatives

Y Liu, M Wang, Y Xu, Y Wu, B Fu, J Li… - Journal of …, 2022 - Wiley Online Library
In order to discover new pesticides with novel modes of action and further study the
sulfoximine scaffolds, 30 novel sulfoximine derivatives were designed, synthesized, and …

Design, synthesis, and structure–activity relationship of quinazolinone derivatives as potential fungicides

JW Peng, XD Yin, H Li, KY Ma, ZJ Zhang… - Journal of Agricultural …, 2021 - ACS Publications
Plant diseases caused by phytopathogenic fungi reduce the yield and quality of crops. To
develop novel antifungal agents, we designed and synthesized eight series of …

Synthesis, fungicidal activity and SAR of 3, 4-dichloroisothiazole-based cycloalkylsulfonamides

Y Zhang, M Wang, M Ahmed, L He, M Ji, Z Qi… - Bioorganic & Medicinal …, 2019 - Elsevier
To develop more valuable and effective fungicide candidates, a novel series of 3, 4-
dichloroisothioxazole-based cycloalkylsulfonamides were synthesized and their structures …

Design, synthesis and fungicidal activities evaluation of N-(thiazol-4-ylmethyl) benzenesulfonamide derivatives

S Zheng, D Huang - Chemical Papers, 2023 - Springer
A series of N-(thiazol-4-ylmethyl) benzenesulfonamide derivatives were designed,
synthesized, and characterized by 1H NMR, 13C NMR, and HRMS. The evaluation of …

Design, Synthesis and Structure-Activity Relationship of Novel Pinacolone Sulfonamide Derivatives against Botrytis cinerea as Potent Antifungal Agents

C Liu, X Xiang, Y Wan, J Yang, Y Li, X Zhang, Z Qi… - Molecules, 2022 - mdpi.com
To develop new fungicides with high efficiency, 46 novel sulfonamide derivatives were
designed and synthesized by introducing pinacolone fragment into chesulfamide which was …

Synthesis, Antifungal, and Antibacterial Activities of Novel Benzoylurea Derivatives Containing a Pyrimidine Moiety

J An, W Lan, Q Fei, P Li, W Wu - Molecules, 2023 - mdpi.com
To explore more efficient and less toxic antibacterial and antifungal pesticides, we utilized 2,
6-difluorobenzamide as a starting material and ultimately synthesized 23 novel benzoylurea …

Sulfonate derivatives bearing an amide unit: design, synthesis and biological activity studies

Y Liu, C Li, M Nie, F Wang, X Ren, L Jin, X Zhou - BMC chemistry, 2024 - Springer
Pest disasters which occurs on crops is a serious problem that not only cause crop yield loss
or even crop failure but can also spread a number of plant diseases. Sulfonate derivatives …