Alkaloids from Eschscholzia californica and Their Capacity to Inhibit Binding of [3H]8-Hydroxy-2-(di-N-propylamino)tetralin to 5-HT1A Receptors in Vitro
S Gafner, BM Dietz, KL McPhail, IM Scott… - Journal of natural …, 2006 - ACS Publications
A 70% ethanol extract of California poppy (Eschscholzia californica) was able to bind to 5-
HT1A and 5-HT7 receptors at 100 μg/mL. The subsequent isolation procedure yielded the …
HT1A and 5-HT7 receptors at 100 μg/mL. The subsequent isolation procedure yielded the …
The active principles of the branchlet and hook of Uncaria sinensis Oliv. examined with a 5-hydroxytryptamine receptor binding assay
H Kanatani, H Kohda, K Yamasaki… - Journal of Pharmacy …, 1985 - academic.oup.com
Of the alkaloids obtained from Uncaria sinensis Oliv., geissoschizine methyl ether,
corynantheine and dihydrocorynantheine decreased specific [3H] 5-HT binding to …
corynantheine and dihydrocorynantheine decreased specific [3H] 5-HT binding to …
Semisynthetic Studies on and Biological Evaluation of N-Methyllaurotetanine Analogues as Ligands for 5-HT Receptors
S Madapa, WW Harding - Journal of Natural Products, 2015 - ACS Publications
N-Methyllaurotetanine (1) has been reported to display good affinity for the 5-HT1A receptor,
but no structure–affinity studies have been performed to date. The commercially available …
but no structure–affinity studies have been performed to date. The commercially available …
Screening of medicinal plants from Suriname for 5-HT1A ligands: Bioactive isoquinoline alkaloids from the fruit of Annona muricata
JA Hasrat, L Pieters, JP De Backer, G Vauquelin… - Phytomedicine, 1997 - Elsevier
Plants from Suriname (South-America) and several Annona species, including A. muricata,
A. ckerimolia, A. montana and A. glabra were screened for 5-HT1A receptor binding activity …
A. ckerimolia, A. montana and A. glabra were screened for 5-HT1A receptor binding activity …
Purpurascenines A–C, Azepino-Indole Alkaloids from Cortinarius purpurascens: Isolation, Biosynthesis, and Activity Studies on the 5-HT2A Receptor
Three previously undescribed azepino-indole alkaloids, named purpurascenines A–C (1–3),
together with the new-to-nature 7-hydroxytryptophan (4) as well as two known compounds …
together with the new-to-nature 7-hydroxytryptophan (4) as well as two known compounds …
5‐Hydroxytryptamine2A receptor binding activity of compounds from Litsea sessilis
LY Chung, MW Lo, MR Mustafa… - … Journal Devoted to …, 2009 - Wiley Online Library
A 96‐well microplate filtration based 5‐HT2A receptor‐radioligand binding assay was
optimized and adopted to carry out a bioassay‐guided fractionation of the methanol extract …
optimized and adopted to carry out a bioassay‐guided fractionation of the methanol extract …
Effects of Geissoschizine Methyl Ether, an Indole Alkaloid in Uncaria Hook, a Constituent of Yokukansan, on Human Recombinant Serotonin7 Receptor
T Ueki, A Nishi, S Imamura, H Kanno… - Cellular and molecular …, 2013 - Springer
Abstract Effects of seven alkaloids, geissoschizine methyl ether (GM), hirsutine, hirsuteine,
rhynchophylline, isorhynchophylline, corynoxeine and isocorynoxeine, in Uncaria hook, a …
rhynchophylline, isorhynchophylline, corynoxeine and isocorynoxeine, in Uncaria hook, a …
Activity of Parthenolide at 5HT2A Receptors
JT Weber, MF O'Connor, K Hayataka… - Journal of natural …, 1997 - ACS Publications
Parthenolide displaces [3H] ketanserin from 5HT2A receptors from rat and rabbit brain and
cloned 5HT2A receptors. K i's are in the 100− 250 μM range. These results suggest that …
cloned 5HT2A receptors. K i's are in the 100− 250 μM range. These results suggest that …
Partial agonistic effect of yokukansan on human recombinant serotonin 1A receptors expressed in the membranes of Chinese hamster ovary cells
K Terawaki, Y Ikarashi, K Sekiguchi, Y Nakai… - Journal of …, 2010 - Elsevier
ETHNOPHARMACOLOGICAL RELEVANCE: Yokukansan (YKS) is a traditional Japanese
medicine consisted of seven medicinal herbs and has been used for treatment of neurosis …
medicine consisted of seven medicinal herbs and has been used for treatment of neurosis …
Stilbene derivatives as human 5-HT6 receptor antagonists from the root of Caragana sinica
MATERIALS AND METHODS Plant Materials The root of C. sinica was collected at
Changnyeong-gun, Gyeongsangnam-do, Korea in July 1995 and the plant was identified by …
Changnyeong-gun, Gyeongsangnam-do, Korea in July 1995 and the plant was identified by …