The 5‐HT1A receptor affinities and ionization constants of a set of 1‐arylpiperazine (4) 1, 2,
3, 4‐tetrahydroisoquinoline (6), and‐quinoline (7) containing N‐(ω‐arylalkyl) or N‐(E) …

A series of 4-amino-5-chloro-2-methoxybenzoates and benzamides containing the 5-and 6-
isoquinuclidinyl system was synthesised and evaluated for binding to 5-HT3, 5-HT4 and D2 …

A novel (4, 5-dihydroimidazol-2-yl)-biphenylamine series of 5-HT7 agonist compounds was
developed from a structurally related lead compound 1. The newly discovered series is …

Phenylpyrroles, a new chemolibrary virtual screening class of 5-HT7 receptor ligands -
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Publisher Summary This chapter discusses taxonomy, indole alkaloids from chemically
investigated Tabernaemontana species, structure elucidation and chemistry, and …

Phytochemical investigations of Terminalia arjuna bark and Terminalia chebula fruits
resulted in the isolation of twelve triterpenoids including two new oleanane type triterpene …

1 Two novel selective 5‐HT6 receptor ligands E‐6801 (6‐chloro‐N‐(3‐(2‐(dimethylamino)
ethyl)‐1H‐indol‐5‐yl) imidazo [2, 1‐b] thiazole‐5‐sulfonamide) and E‐6837 (5‐chloro‐N‐(3 …

The preparation of a novel class of 4-(2-aminoethoxy)-N-(phenylsulfonyl) indoles which
exhibit high affinity towards the 5-HT6 receptor is reported here. Among these compounds, 4 …

Chemical analysis of Atriplex halimus (Family: Chenopodiaceae) revealed that the plant at
Wadi-Hof and Wadi-Sudr habitats contained eleven free amino acids with different range of …

1 Skimmianine, kokusaginine and confusameline, three furoquinolines extracted from the
leaves of Evodia merrillii (Rutaceae), were investigated to characterize their selective effects …