Botrytis cinerea is an economically important fungal pathogen with a host range of over 200
plant species. Unfortunately, gray mold disease caused by B. cinerea has not been …

Starting from the key intermediate 5-(3, 4, 5-trimethoxyphenyl)-1, 3, 4-thiadiazole-2-thiol (4)
or the oxadiazole analogue (5), the title compounds 9 and 10 are synthesized by a two-step …

Plant fungal diseases have caused great decreases in crop quality and yield. As one of the
considerable agricultural diseases, cucumber downy mildew (CDM) caused by …

In order to rapidly prepare novel lead compounds of fungicides, the method that involved
both the combinatorial chemistry and the conventional synthesis was used. The fungicidal …

BACKGROUND: With the objective of exploring the fungicidal activity of 2‐
oxocyclohexylsulfonamides (2), a series of novel 2‐amino‐6‐oxocyclohexenylsulfonamides …

Sulfone derivatives, an important synthetic strategy in drug discovery, are acquiring more
importance in plant protection field in recent years because of their pesticide activities, such …

A series of novel ethyl 4‐(methyl or trifluoromethyl)‐2‐(2‐(substituted phenoxy) acetamido)
thiazole‐5‐carboxylates 7a, 7b, 7c, 7d, 7e and 8f, 8g, 8h, 8i, 8j, 8k, 8l, 8m, 8n, 8o, 8p, 8q, 8r …

A series of structurally novel 1, 3, 4-oxadiazole thioether derivatives (6a–6z) containing a 6-
fluoroquinazolinylpiperidinyl moiety were designed and synthesized using pharmacophore …

Acetohydroxyacid synthase (AHAS) was considered as a promising target for antifungal
agents. Herein, three series of novel sulfonylureas (SUs) 9− 11 containing aromatic …

As a part of our continuing exploration to discover new potential promising fungicide
candidates, eighteen sulfonate derivatives (3a–3r) containing a kakuol moiety were …