Synthesis, biological activity and three-dimensional quantitative structure-activity relationship (3D-QSAR) study of novel 4-methyl-1, 2, 4-triazole-thioethers containing …

Y Yu, W Duan, G Lin, G Kang, X Wang… - Chinese Journal of …, 2020 - sioc-journal.cn
A series of novel 4-methyl-1, 2, 4-triazole-thioethers containing gem-dimethylcyclopropane
ring were designed and synthesized by multi-step reactions in search of potent novel …

Design, synthesis, and fungicidal evaluation of a series of novel 5-methyl-1H-1, 2, 3-trizole-4-carboxyl amide and ester analogues

ZJ Wang, Y Gao, YL Hou, C Zhang, SJ Yu… - European Journal of …, 2014 - Elsevier
Succinate dehydrogenase inhibitors (SDHIs) are efficient fungicides that are widely used to
control plant diseases caused by phytopathogenic fungi, although their effectiveness is …

[HTML][HTML] Design, Synthesis, and Antifungal Activity of Some Novel Phenylthiazole Derivatives Containing an Acylhydrazone Moiety

Y Tian, J Shi, X Deng, T Yu, Y Hu, R Hu, Y Lei, L Yu… - Molecules, 2023 - mdpi.com
Crop fungal diseases pose a serious threat to global crop production and quality.
Developing new and efficient fungicides is an important measure to control crop diseases …

[HTML][HTML] Design, Synthesis and Biological Evaluation of N-((2-phenyloxazol-4-yl)methyl) Pyrimidine Carboxamide Derivatives as Potential Fungicidal Agents

D Huang, S Zheng, YX Cheng - Heterocyclic Communications, 2020 - degruyter.com
Abstract Twelve N-((2-phenyloxazol-4-yl) methyl) pyrimidine carboxamide derivatives were
designed, synthesized, and characterized by 1H NMR, 13C NMR, and HRMS. The …

[HTML][HTML] Sulfonate derivatives bearing an amide unit: design, synthesis and biological activity studies

Y Liu, C Li, M Nie, F Wang, X Ren, L Jin, X Zhou - BMC chemistry, 2024 - Springer
Pest disasters which occurs on crops is a serious problem that not only cause crop yield loss
or even crop failure but can also spread a number of plant diseases. Sulfonate derivatives …

Synthesis and fungicidal activity of 2-oxocyclohexylsulfonamides containing fluorine

Y Hong-ye, YAN Xiao-jing, Y Hui-zhu… - Chinese Journal of …, 2010 - nyxxb.cn
Nine novel 2-oxocyclohexylsulfonamides containing fluorine were synthesized from
cyclohexanone and their structures were confirmed by 1H NMR, 13C NMR and elemental …

Design, synthesis and SAR study of novel sulfonylureas containing an alkenyl moiety

W Wei, D Cheng, J Liu, Y Li, Y Ma, Y Li, S Yu… - Organic & …, 2016 - pubs.rsc.org
A series of sulfonylurea compounds was designed and synthesized via introducing an
alkenyl moiety into the aryl-5 position and most title compounds exhibited enhanced …

Novel sulfone derivatives containing a 1, 3, 4‐oxadiazole moiety: design and synthesis based on the 3D‐QSAR model as potential antibacterial agent

J Chen, Y Luo, C Wei, S Wu, R Wu… - Pest management …, 2020 - Wiley Online Library
BACKGROUND The rice bacterial leaf blight (BLB) is one of the most serious bacterial
diseases caused by Xanthomonas oryzae pv. oryzae (Xoo), which can cause yield loss of …

Design, Synthesis, Antifungal Activities and SARs of (R)‐2‐Aryl‐4,5‐dihydrothiazole‐4‐carboxylic Acid Derivatives

J Liu, Y Li, Y Chen, X Hua, Y Wan… - Chinese Journal of …, 2015 - Wiley Online Library
Based on the structure of natural product 2‐aryl‐4, 5‐dihydrothiazole‐4‐carboxylic acid, a
series of novel (R)‐2‐aryl‐4, 5‐dihydrothiazole‐4‐carboxylic acid derivatives were designed …

[HTML][HTML] Novel 1, 3, 4-oxadiazole thioether and sulfone derivatives bearing a flexible N-heterocyclic moiety: Synthesis, characterization, and anti-microorganism …

F Wang, BX Yang, TH Zhang, QQ Tao, X Zhou… - Arabian Journal of …, 2023 - Elsevier
In the search for more efficient and versatile anti-phytopathogen agents, a series of new 1, 3,
4-oxadiazole thioether/sulfone analogues bearing a flexible N-containing heterocyclic …