Synthesis and Antifungal Activity of 2-Substituted Sulfinyl (Sul-fonyl)-5-(4-nitro or 4-methoxyphenyl)-1, 3, 4-thiadiazole Derivatives

C Yang, S Yang, BA SONG, DY HU… - Chinese Journal of …, 2010 - sioc-journal.cn
Starting from p-nitrobenzoic acid and p-methoxybenzoic acid, seven new 2-sub-stitutedthio-
5-(4-nitro or 4-methoxyphenyl)-1, 3, 4-thiadiazole compounds 5 were synthesized in five …

Synthesis of benzothiazole-appended bis-triazole-based structural isomers with promising antifungal activity against Rhizoctonia solani

RK Upadhyay, KK Saini, N Deswal, T Singh… - RSC …, 2022 - pubs.rsc.org
In order to explore new antifungal agrochemicals, we reported the synthesis of two series 5a–
f, 6 and 7a–f, 8 of benzothiazole-appended bis-triazole derivative-based structural isomers …

Novel 5-chloro-pyrazole derivatives containing a phenylhydrazone moiety as potent antifungal agents: synthesis, crystal structure, biological evaluation and a 3D …

J Jiao, A Wang, M Chen, MQ Wang… - New Journal of Chemistry, 2019 - pubs.rsc.org
Based on the active substructure combination principle, twenty-four novel 5-chloro-pyrazole
derivatives containing a phenylhydrazone moiety were designed, synthesized, and …

Synthesis, antifungal activity and molecular docking study of 1, 3, 4-thiadiazole-urea compounds containing gem-dimethylcyclopropane ring structure

C Yucheng, C Meihua, L Guishan… - Chinese Journal of …, 2022 - sioc-journal.cn
In an attempt to search for natural renewable product-based antifungal agents, eighteen 1,
3, 4-thiadiazole-urea compounds containing gem-dimethylcyclopropane ring structure were …

Synthesis of pyrazole-4-carboxamides as potential fungicide candidates

C Dong, W Gao, X Li, S Sun, J Huo, Y Wang, D Ren… - Molecular Diversity, 2021 - Springer
A series of novel pyrazole-4-carboxamides were rationally designed, synthesized, and their
structures were characterized by 1 H NMR, 13 C NMR and HRMS. Preliminary bioassay …

Synthesis and anti-phytopathogenic activity of 8-hydroxyquinoline derivatives

XD Yin, Y Sun, RK Lawoe, GZ Yang, YQ Liu… - RSC …, 2019 - pubs.rsc.org
Phytopathogenic fungi have become a serious threat to the quality of agricultural products,
food security and human health globally, necessitating the need to discover new antifungal …

Synthesis, biological activities and 3D-QSAR studies of (R)-2-phenyl-4, 5-dihydrothiazole-4-carboxamide derivatives containing a sulfur ether moiety

J Liu, F Li, Y Wang, H Zhang, J Dong, P Sun, Y Li… - Chinese Chemical …, 2019 - Elsevier
Abstract A series of (R)-2-phenyl-4, 5-dihydrothiazole-4-carboxamide derivatives containing
a sulfur ether moiety were synthesized and characterized on the basis of NMR and …

Synthesis and fungicidal activity of novel 2-aryl-3-(1, 3, 4-thiadiazolyl)-6 (8)-methyl-1, 3-benzoxazines

Z Tang, Z Xia, S Chang, Z Wang - Bioorganic & medicinal chemistry letters, 2015 - Elsevier
A class of novel 2-aryl-3-(1, 3, 4-thiadiazolyl)-6 (8)-methyl-1, 3-benzoxazines was prepared
by reactions of 2-methyl-6-((1, 3, 4-thiadiazolylamino) methyl) phenols or 4-methyl-2-((1, 3, 4 …

Design and synthesis of novel cylopentapyrazoles bearing 1, 2, 3-thiadiazole moiety as potent antifungal agents

B Giray, AE Karadağ, ÖŞ İpek, H Pekel, M Güzel… - Bioorganic …, 2020 - Elsevier
In drug-resistant phytopathogenic fungi, there has been extensive research on
microbiological and antifungal drug development. In this study, a novel series of …

Novel trifluoromethylpyrazole acyl thiourea derivatives: synthesis, antifungal activity and docking study

H Wang, ZW Zhai, YX Shi, CX Tan… - Letters in Drug …, 2019 - ingentaconnect.com
Background: In recent years, pyrazole carboxamide derivatives possessed excellent
fungicidal activity. In the process of designing new fungicides, the carboxamide group was …