Synthesis and biological evaluation of substituted phenyl azetidine-2-one sulphonyl derivatives as potential antimicrobial and antiviral agents

MK Mandal, S Ghosh, HR Bhat, L Naesens… - Bioorganic …, 2020 - Elsevier
In the present study, we intend to synthesize a series of novel substituted phenyl azetidine-2-
one sulphonyl derivatives. The entire set of derivatives 5 (at) were screened for in-vitro …

Synthesis, In Vitro Evaluation, and Molecular Docking Studies of Azetidinones and Thiazolidinones of 2‐Amino‐5‐cyclopropyl‐1,3,4‐thiadiazole as Antibacterial …

H Patel, L Mishra, M Noolvi, R Karpoormath… - Archiv der …, 2014 - Wiley Online Library
In an attempt to find a new class of antimicrobial agents, a series of novel azetidin‐2‐ones
3a–e and thiazolidin‐4‐ones 4a–e of 2‐amino‐5‐cyclopropyl‐1, 3, 4‐thiadiazole were …

[HTML][HTML] Synthesis and antimicrobial activity of new pyridine containing substituted phenyl azetidine-2-one derivatives

VE Rani, PR Reddy - Open Journal of Medicinal Chemistry, 2018 - scirp.org
The most important nitrogen containing heterocycles of pyridine containing substituted
phenyl azetidine-2-ones have found pharmacological application such as antibiotics and …

Synthesis and antimicrobial activity of new tetrahydro‐naphthalene‐thiazolidinedione and thiohydantoine derivatives

Z Ates‐Alagoz, N Altanlar… - Journal of Heterocyclic …, 2009 - Wiley Online Library
As part of an ongoing program aimed at recognizing novel antioxidant, antimicrobial, and
anticancer molecules, herein we report the synthesis and biological evaluation of …

Novel N-Substituted 3-Aryl-4-(diethoxyphosphoryl) azetidin-2-ones as antibiotic enhancers and antiviral agents in search for a successful treatment of complex …

IE Głowacka, M Grabkowska-Drużyc, G Andrei… - International Journal of …, 2021 - mdpi.com
A novel series of N-substituted cis-and trans-3-aryl-4-(diethoxyphosphoryl) azetidin-2-ones
were synthesized by the Kinugasa reaction of N-methyl-or N-benzyl-(diethyoxyphosphoryl) …

Synthesis, antimicrobial and antiviral evaluation of substituted imidazole derivatives

D Sharma, B Narasimhan, P Kumar, V Judge… - European journal of …, 2009 - Elsevier
In the present study, we have synthesized 2-(substituted phenyl)-1H-imidazole (1–12) and
(substituted phenyl)-[2-(substituted phenyl)-imidazol-1-yl]-methanone (13–26) analogues …

Synthesis and antimicrobial activity of some amide derivatives bearing thiazole, benzhydryl and piperidine moieties

A Ozdemir - Letters in Drug Design & Discovery, 2013 - ingentaconnect.com
In the present study, N-(benzhydryl/thiazol-2-yl)-2-(piperidin-1-yl) acetamide derivatives
were obtained by the reaction of 2-chloro-N-(benzhydryl/thiazole-2-yl) acetamides with …

Facile synthesis, antimicrobial and antiviral evaluation of novel substituted phenyl 1, 3-thiazolidin-4-one sulfonyl derivatives

MK Mandal, S Ghosh, L Naesens, HR Bhat… - Bioorganic …, 2021 - Elsevier
A series of novel substituted phenyl 1, 3-thiazolidin-4-one sulfonyl derivatives 5 (at) were
synthesized and screened for their in-vitro anti-microbial and anti-viral activity. The result of …

[HTML][HTML] Synthesis, characterization, biological evaluation and docking studies of novel 5-(2-methyl-1, 8-naphthyridin-3-yl)-1, 3, 4-oxadiazol-2-amine and some of its …

RK Parangi, R Domala - Results in Chemistry, 2023 - Elsevier
The present work demonstrates the novel compounds of 5-(2-methyl-1, 8-naphthyridin-3-yl)-
1, 3, 4-oxadiazol-2-amine and its derivatives using symmetrical anhydrides. The synthesized …

Synthesis, characterization, and antimicrobial activity of new thienopyrimidine derivatives

M Ahmed, M Sayed, AF Saber… - Polycyclic Aromatic …, 2022 - Taylor & Francis
Nowadays heterocyclic compounds containing pyrimidine scaffold attract the interest of
many organic chemists due to their strong biological activity, so herein we present the …