Synthesis of novel antibacterial and antifungal quinoxaline derivatives

X Tang, Q Zhou, W Zhan, D Hu, R Zhou, N Sun… - RSC …, 2022 - pubs.rsc.org
A series of quinoxaline derivatives were designed, synthesized and evaluated as
antimicrobial agents against plant pathogenic bacteria and fungi. Some of these compounds …

Design, synthesis, and structure–activity relationship of quinazolinone derivatives as potential fungicides

JW Peng, XD Yin, H Li, KY Ma, ZJ Zhang… - Journal of Agricultural …, 2021 - ACS Publications
Plant diseases caused by phytopathogenic fungi reduce the yield and quality of crops. To
develop novel antifungal agents, we designed and synthesized eight series of …

Design, Synthesis, Antifungal, and Antioxidant Activities of (E)-6-((2-Phenylhydrazono)methyl)quinoxaline Derivatives

M Zhang, ZC Dai, SS Qian, JY Liu, Y Xiao… - Journal of agricultural …, 2014 - ACS Publications
Different substituted phenylhydrazone groups were linked to the quinoxaline scaffold to
provide 26 compounds (6a–6z). Their structures were confirmed by 1H and 13C NMR, MS …

Synthesis and anti-phytopathogenic activity of 8-hydroxyquinoline derivatives

XD Yin, Y Sun, RK Lawoe, GZ Yang, YQ Liu… - RSC …, 2019 - pubs.rsc.org
Phytopathogenic fungi have become a serious threat to the quality of agricultural products,
food security and human health globally, necessitating the need to discover new antifungal …

Synthesis and pesticidal activities of new quinoxalines

XH Liu, W Yu, LJ Min, DE Wedge, CX Tan… - Journal of Agricultural …, 2020 - ACS Publications
Natural products are a source of many novel compounds with biological activity for the
discovery of new pesticides and pharmaceuticals. Quinoxaline is a fused N-heterocycle in …

Design, Synthesis, Antibacterial Evaluation, Three-Dimensional Quantitative Structure–Activity Relationship, and Mechanism of Novel Quinazolinone Derivatives

L Shao, S Zhao, S Yang, X Zhou, Y Li, C Li… - Journal of Agricultural …, 2023 - ACS Publications
Plant bacterial illnesses are common and cause dramatic damage to agricultural goods all
over the world, yet there are few efficient bactericides to alleviate them at present. To …

Design, Synthesis, and Biological Evaluation of Novel Thiazolidinone-Containing Quinoxaline-1,4-di-N-oxides as Antimycobacterial and Antifungal Agents

H Zhang, J Zhang, W Qu, S Xie, L Huang… - Frontiers in …, 2020 - frontiersin.org
Tuberculosis and fungal infections can pose serious threats to human health. In order to find
novel antimicrobial agents, 26 novel quinoxaline-1, 4-di-N-oxides containing a …

Novel vanillin derivatives containing a 1, 3, 4-thiadiazole moiety as potential antibacterial agents

Q Wu, H Cai, T Yuan, S Li, X Gan, B Song - Bioorganic & medicinal …, 2020 - Elsevier
In this study, thirty-four novel vanillin derivatives containing a 1, 3, 4-thiadiazole structure
were obtained and their antibacterial activities were evaluated. The results indicate that most …

Design and discovery of novel antifungal quinoline derivatives with acylhydrazide as a promising pharmacophore

YD Yang, YH He, KY Ma, H Li, ZJ Zhang… - Journal of Agricultural …, 2021 - ACS Publications
Inspired by natural 2-quinolinecarboxylic acid derivatives, a series of quinoline compounds
containing acylhydrazine, acylhydrazone, sulfonylhydrazine, oxadiazole, thiadiazole, or …

Design, synthesis, and evaluation of new sulfone derivatives containing a 1, 3, 4-oxadiazole moiety as active antibacterial agents

P Li, D Hu, D Xie, J Chen, L Jin… - Journal of agricultural and …, 2018 - ACS Publications
This study aimed to synthesize some new sulfone derivatives containing a 1, 3, 4-oxadiazole
moiety and investigate their in vitro antibacterial activities against Xanthomonas oryzae pv …