Novel pyrimidine derivatives bearing a 1, 3, 4-thiadiazole skeleton: Design, synthesis, and antifungal activity

N Pan, C Liu, R Wu, Q Fei, W Wu - Frontiers in Chemistry, 2022 - frontiersin.org
In this study, twenty novel pyrimidine derivatives bearing a 1, 3, 4-thiadiazole skeleton were
designed and synthesized. Then their antifungal activity against Botrytis cinereal (B …

Synthesis and antifungal activity of pyrimidine derivatives containing an amide moiety

W Wu, W Lan, C Wu, Q Fei - Frontiers in chemistry, 2021 - frontiersin.org
In this study, 17 novel pyrimidine derivatives containing an amide moiety were synthesized.
Then their in vitro antifungal activities against Botryosphaeria dothidea (B. dothidea) …

A facile green synthesis and in vitro antimicrobial activity 4H-pyrimido [2, 1-b][1, 3] benzothiazole derivatives using aluminum trichloride under solvent free conditions

PK Sahu, PK Sahu, J Lal, D Thavaselvam… - Medicinal Chemistry …, 2012 - Springer
Aluminum trichloride acts as readily available, inexpensive, and efficient catalyst for one-pot
three-component condensation reaction of aldehydes, dicarbonyl, and 2-amino …

Synthesis and fungicidal activity of novel 1, 2, 4-triazole derivatives containing a pyrimidine moiety

WN Wu, YM Jiang, Q Fei, HT Du - Phosphorus, Sulfur, and Silicon …, 2019 - Taylor & Francis
Abstract A series of novel 1, 2, 4-triazole derivatives containing a pyrimidine moiety were
synthesized and their fungicidal activities were evaluated. The preliminary biological test …

Synthesis and bioactivities study of novel pyridylpyrazol amide derivatives containing pyrimidine motifs

W Wu, M Chen, Q Fei, Y Ge, Y Zhu, H Chen… - Frontiers in …, 2020 - frontiersin.org
In this study, thirteen new pyridylpyrazolamide derivatives containing pyrimidine motifs were
synthesized via six-step reactions. Bioassay results showed that some of the synthesized …

Novel pyrimidine derivatives containing an amide moiety: design, synthesis, and antifungal activity

W Wu, M Chen, R Wang, H Tu, M Yang, G Ouyang - Chemical Papers, 2019 - Springer
The objectives of the current study were to synthesize a series of novel pyrimidine
derivatives containing an amide moiety and to investigate their in vitro antifungal activities …

Design, synthesis, antibacterial, and antifungal evaluation of phenylthiazole derivatives containing a 1, 3, 4-thiadiazole thione moiety

G Mao, Y Tian, J Shi, C Liao, W Huang, Y Wu, Z Wen… - Molecules, 2024 - mdpi.com
To effectively control the infection of plant pathogens, we designed and synthesized a series
of phenylthiazole derivatives containing a 1, 3, 4-thiadiazole thione moiety and screened for …

Design, synthesis and antimicrobial activities of novel 1, 3, 5-thiadiazine-2-thione derivatives containing a 1, 3, 4-thiadiazole group

J Yan, W Si, H Hu, X Zhao, M Chen, X Wang - PeerJ, 2019 - peerj.com
A series of novel 1, 3, 5-thiadiazine-2-thione derivatives containing a 1, 3, 4-thiadiazole
group was designed and synthesized. The structures of all the compounds were well …

Synthesis and fungicidal activity of novel 2, 5-disubstituted-1, 3, 4-thiadiazole derivatives containing 5-phenyl-2-furan

ZN Cui, YS Li, DK Hu, H Tian, JZ Jiang, Y Wang… - Scientific Reports, 2016 - nature.com
Abstract A series of 2, 5-disubstituted-1, 3, 4-thiadiazoles were synthesized using
Lawesson's reagent by an efficient approach under microwave irradiation in good yields …

Synthesis and antimicrobical evaluation of a novel class of 1, 3, 4-thiadiazole: derivatives bearing 1, 2, 4-triazolo [1, 5-a] pyrimidine moiety

Y Luo, S Zhang, ZJ Liu, W Chen, J Fu, QF Zeng… - European journal of …, 2013 - Elsevier
A series of novel 1, 3, 4-thiadiazole derivatives bearing 1, 2, 4-triazolo [1, 5-a] pyrimidine
moiety were synthesized by the method of splicing active substructures. Among these …