Design, synthesis and bioactivity of novel 2-aryl-4-alkylthiazole-5-carboxylic acid derivatives

Y Zhu, D Wang, Y Yuan, Y Ma, X Zou… - Chinese Journal of …, 2012 - sioc-journal.cn
To find new lead compounds with muti-bioactivities, a series of novel 1, 3-thiazole-5-
carboxylic acid derivatives containing aryloxyacetate were designed via the method of …

Synthesis and Biological Activities of 1, 2, 3-Thiadiazole Derivatives Containing 1, 3, 4-Thiadiazole Moiety

S Wang, X Zuo, Z Fan, Z Zhang, J Zhang… - Chinese Journal of …, 2013 - sioc-journal.cn
To find novel pesticide lead compounds with highly active bioactivity, 32 novel 1, 2, 3-
thiadiazole derivatives con-taining 1, 3, 4-thiadiazole ring were designed and synthesized …

Design, Synthesis, Antifungal Activities and SARs of (R)‐2‐Aryl‐4,5‐dihydrothiazole‐4‐carboxylic Acid Derivatives

J Liu, Y Li, Y Chen, X Hua, Y Wan… - Chinese Journal of …, 2015 - Wiley Online Library
Based on the structure of natural product 2‐aryl‐4, 5‐dihydrothiazole‐4‐carboxylic acid, a
series of novel (R)‐2‐aryl‐4, 5‐dihydrothiazole‐4‐carboxylic acid derivatives were designed …

Synthesis and biological activities of thio-triazole derivatives as novel potential antibacterial and antifungal agents

QP Wang, JQ Zhang, GLV Damu, K Wan… - Science China …, 2012 - Springer
A series of novel thio-triazole derivatives including thiols, thioethers and thiones as well as
some corresponding triazolium compounds were conveniently and efficiently synthesized …

Synthesis, Structure and Biological Activities of1, 3-Thiazolidine Derivatives

JQ Weng, DL Shen, CX Tan - Chinese Journal of Organic Chemistry, 2006 - sioc-journal.cn
In order to find new thiazole-heterocycle lead compounds, six 2-oxo/thio-1, 3-thiazolidine-3-
carboxylates 3 and five N-substituted benzoyl-2-oxo/thio-1, 3-thiazolidines 5 were …

Synthesis and antifungal activities of N-1, 3, 4-thiadiazol-2-yl-4-oxo-thiochroman-2-yl-formamide derivatives

XY Han, SB Li, GC Liang, G Zhou… - Yao xue xue bao …, 2017 - europepmc.org
Thiochromanones and 1, 3, 4-thiadiazoles as heterocyclic compounds have broad
biological activities. In order to find novel compounds with antifungal bioactivity, substituted …

Synthesis, Structure, and Biological Activity of Novel 1H‐1,2,4‐Triazol‐1‐yl‐thiazole Derivatives

S Ling, Z Xin, Z Qing, L Jian‐Bing, J Zhong… - Synthetic …, 2007 - Taylor & Francis
Amino‐4‐aryl‐5‐(1 H‐1, 2, 4‐triazol‐1‐yl) thiazole derivatives were synthesized from the
reaction of α‐bromo substituted acetophenone and thiourea. The structures were confirmed …

Syntheses and biological activities of novel benzotriazole compounds containing a thioamide group

L XU, Z ZHAI, G YU, Y QIN, Y YANG - Chemical Research in Chinese …, 2006 - Elsevier
(E)-2-(1H-Benzo [d][1, 2, 3] triazol-1-yl)-3-(4-chlorophenyl)-3-hydroxy-N-phenylprop-2-
enethioamide (compound 1) and (E)-2-(1H-benzo [d][1, 2, 3] triazol-1-yl)-3-hydroxy-N, 3 …

Synthesis, structure and biological activities of N-arylaminocarbonyl-2-oxo/thio-thiazolidine

JQ Weng, DL Shen, CX Tan, XM Ou - Chinese Journal of Organic …, 2006 - sioc-journal.cn
In order to find new thiazole-heterocycle lead compounds, seventeen N-arylaminocarbonyl-
2-oxo/thio-thiazolidine derivatives were synthesized from a coupling reaction of 2-oxo/thio …

Synthesis and Antifungal Activity of 2-Substituted Sulfinyl (Sul-fonyl)-5-(4-nitro or 4-methoxyphenyl)-1, 3, 4-thiadiazole Derivatives

C Yang, S Yang, BA SONG, DY HU… - Chinese Journal of …, 2010 - sioc-journal.cn
Starting from p-nitrobenzoic acid and p-methoxybenzoic acid, seven new 2-sub-stitutedthio-
5-(4-nitro or 4-methoxyphenyl)-1, 3, 4-thiadiazole compounds 5 were synthesized in five …