Thiazole-containing compounds as therapeutic targets for cancer therapy
In the last few decades, considerable progress has been made in anticancer agents
development, and several new anticancer agents of natural and synthetic origin have been …
development, and several new anticancer agents of natural and synthetic origin have been …
Anticancer potential of thiazole derivatives: a retrospective review
S Jain, S Pattnaik, K Pathak, S Kumar… - Mini reviews in …, 2018 - ingentaconnect.com
This review brings forth the potential of thiazole derivatives for their anticancer activities. The
emphasis is placed on the structural diversity of thiazole derivatives, responsible for their …
emphasis is placed on the structural diversity of thiazole derivatives, responsible for their …
[HTML][HTML] Thiazole ring-the antimicrobial, anti-inflammatory, and anticancer active scaffold
S Hosseininezhad, A Ramazani - Arabian Journal of Chemistry, 2023 - Elsevier
Background Thiazole ring is one of the most important heterocycle scaffolds in organic and
medicinal chemistry due to this scaffold being the backbone of numerous drugs and their …
medicinal chemistry due to this scaffold being the backbone of numerous drugs and their …
Synthesis of 2-trifluoromethyl thiazoles via [3+ 2] cycloaddition of pyridinium 1, 4-zwitterionic thiolates with CF 3 CN
Y Yao, B Lin, M Wu, Y Zhang, Y Huang… - Organic & …, 2022 - pubs.rsc.org
2, 2, 2-Trifluoroacetaldehyde O-(aryl) oxime was employed for the [3+ 2] cycloaddition of
pyridinium 1, 4-zwitterionic thiolates for the synthesis of 2-trifluoromethyl 4, 5-disubstituted …
pyridinium 1, 4-zwitterionic thiolates for the synthesis of 2-trifluoromethyl 4, 5-disubstituted …
Antibacterial evaluation and molecular docking studies of pyrazole–thiosemicarbazones and their pyrazole–thiazolidinone conjugates
O Ebenezer, A Singh-Pillay, NA Koorbanally… - Molecular Diversity, 2021 - Springer
A library of pyrazole–thiazolidinone conjugates was synthesized using a molecular
hybridization approach through a Vilsmeier–Haack reaction. The compounds were tested for …
hybridization approach through a Vilsmeier–Haack reaction. The compounds were tested for …
[HTML][HTML] A potential antifungal agent: Insight into the antifungal mechanism against Phomopsis sp
C Yuan, T Zhang, J Tian, T Deng, H Xin, Y Liu… - Arabian Journal of …, 2024 - Elsevier
Abstract 19 myricetin derivatives containing thiazole were designed and synthesized. Their
fungicidal activities in vitro against ten species of plant pathogenic fungi were evaluated …
fungicidal activities in vitro against ten species of plant pathogenic fungi were evaluated …
2, 4, 5-trisubstituted thiazole: A privileged scaffold in drug design and activity improvement
Z Zhang, B Shu, Y Zhang, GS Deora… - Current Topics in …, 2020 - ingentaconnect.com
Thiazole is an important 5-membered heterocyclic compound containing nitrogen and sulfur
atoms with various pharmaceutical applications including anti-inflammatory, anti-cancer, anti …
atoms with various pharmaceutical applications including anti-inflammatory, anti-cancer, anti …
The effect of newly synthesized progesterone derivatives on apoptotic and angiogenic pathway in MCF-7 breast cancer cells
SMM Yahya, AO Abdelhamid, MM Abd-Elhalim… - Steroids, 2017 - Elsevier
Due to its high potency and selectivity, anticancer agents consisting of combined molecules
have gained great interests. The current study introduces newly synthesized progesterone …
have gained great interests. The current study introduces newly synthesized progesterone …
New thiazoline-tetralin derivatives and biological activity evaluation
In this study, novel N′-(3-cyclohexyl/phenyl-4-(substituted phenyl) thiazole-2 (3 H)-ylidene)-
2-[(5, 6, 7, 8-tetrahydronaphthalen-2-yl) oxy] acetohydrazide (4a–4k) derivatives were …
2-[(5, 6, 7, 8-tetrahydronaphthalen-2-yl) oxy] acetohydrazide (4a–4k) derivatives were …
Synthesis, spectral properties and anticancer studies of novel hetrocyclic azo dye ligand derived from 2-amino-5-methyl thiazole with some transition metal complexes
KJ Al-Adilee, HM Hessoon - Journal of Physics: Conference …, 2019 - iopscience.iop.org
This research included preparation of the thiazolyl azo ligand 2-[2--(5-Methyl thiazolyl) azo]-
4-Ethoxy phenol (MeTAEP) and their metal complexes which was prepared by coupling of …
4-Ethoxy phenol (MeTAEP) and their metal complexes which was prepared by coupling of …