Recent progress in cyclic aryliodonium chemistry: syntheses and applications

X Peng, A Rahim, W Peng, F Jiang, Z Gu… - Chemical …, 2023 - ACS Publications
Hypervalent aryliodoumiums are intensively investigated as arylating agents. They are
excellent surrogates to aryl halides, and moreover they exhibit better reactivity, which allows …

Non-coding RNAs in tuberculosis epidemiology: Platforms and approaches for investigating the genome's dark matter

A Almatroudi - International Journal of Molecular Sciences, 2022 - mdpi.com
A growing amount of information about the different types, functions, and roles played by
non-coding RNAs (ncRNAs) is becoming available, as more and more research is done …

Isoflavonoid and furanochromone natural products as potential DNA gyrase inhibitors: Computational, spectral, and antimycobacterial studies

VR Jagatap, I Ahmad, D Sriram, J Kumari, DK Adu… - ACS …, 2023 - ACS Publications
In pursuit of new antitubercular agents, we here report the antimycobacterial (H37Rv) and
DNA gyrase inhibitory potential of daidzein and khellin natural products (NPs). We procured …

New tetrahydropyrimidine-1, 2, 3-triazole clubbed compounds: Antitubercular activity and Thymidine Monophosphate Kinase (TMPKmt) inhibition

MS El-Shoukrofy, A Atta, S Fahmy, D Sriram… - Bioorganic …, 2023 - Elsevier
Two series of new tetrahydropyrimidine (THPM)-1, 2, 3-triazole clubbed compounds were
designed, synthesized and screened for their antitubercular (anti-TB) activity against M …

Combined Bioinformatics and Combinatorial Chemistry Tools to Locate Drug‐Able Anti‐TB Phytochemicals: A Cost‐Effective Platform for Natural Product‐Based Drug …

SS Swain, T Hussain - Chemistry & Biodiversity, 2022 - Wiley Online Library
Based on extensive experimental studies, a huge number of phytochemicals showed
potential activity against tuberculosis (TB) at a lower minimum inhibitory concentration (MIC) …

Synthesis of Indenoquinolinones and 2-Substituted Quinolines via [4 + 2] Cycloaddition Reaction

G Yang, L Yao, G Mao, GJ Deng… - The Journal of Organic …, 2022 - ACS Publications
We have reported a metal-free protocol for the synthesis of indenoquinolinones and 2-
substituted quinolines via [4+ 2] cycloaddition reaction using readily available 2 …

Synthesis of Selenyl-Substituted Quinoline Derivatives via Substrate-Controlled Three-Component Domino Reactions

SS Sun, ZY Mo, YY Chen, YL Xu - The Journal of Organic …, 2022 - ACS Publications
A simple and efficient method for the preparation of selenyl-substituted quinoline derivatives
through a CSp3–H selenylation of in situ-generated 3-acetyl quinoline has been developed …

One-Pot Synthesis of Isoxazole-Fused Tricyclic Quinazoline Alkaloid Derivatives via Intramolecular Cycloaddition of Propargyl-Substituted Methyl Azaarenes under …

Z Wang, Y Zhao, J Chen, M Chen, X Li, T Jiang, F Liu… - Molecules, 2023 - mdpi.com
A practical method was developed for the convenient synthesis of isoxazole-fused tricyclic
quinazoline alkaloids. This procedure accesses diverse isoxazole-fused tricyclic quinazoline …

Coumaryl‐sulfonamide moiety: Unraveling their synthetic strategy and specificity toward hCA IX/XII, facilitating anticancer drug development

M Mahapatra, SK Mekap, S Mal, J Sahoo… - Archiv der …, 2023 - Wiley Online Library
Currently, cancer is the most grieving threat to society. The cancer‐related death rate has
had an ascending trend, despite the implementation of numerous treatment strategies or the …

In Silico Identification of Potential Insect Peptides against Biofilm‐Producing Staphylococcus aureus

A Sahoo, SS Swain, SK Panda, T Hussain… - Chemistry & …, 2022 - Wiley Online Library
Biofilm‐producing Staphylococcus aureus (SA) strains are frequently found in medical
environments, from surgical/wound sites, medical devices. These biofilms reduce the …