Quinazolinones are common substructures in molecules of medicinal importance. We report
an enantioselective copper‐catalyzed borylative cyclization for the assembly of privileged …

Developing novel fungicide candidates are intensively promoted by the rapid emergences of
resistant fungi that outbreak on agricultural production. Aiming to discovery novel antifungal …

2, 3-Dihydroquinazolinone derivatives are known for antiviral, antimicrobial, analgesic, anti-
inflammatory, and anticancer activities. However, recent approaches used for their synthesis …

Axially chiral N‐substituted quinazolinones are important bioactive molecules, which are
presented in many synthetic drugs. However, most strategies toward their atroposelective …

A synthetic method based on radical borylation/cyclization cascades of N-allylcyanamides
was developed to construct diverse boron-substituted N-heterocycles. In the reaction …

A new method for directly synthesizing acylated and alkylated quinazoline derivatives by the
epoxide ring-opening reaction in the presence of I2/DMSO with 2-aminobenzamide is …

Even though several quinazolinone derivatives have been synthesized, still there is a
constant demand for designing and synthesis of new quinazolinone derivatives by fine …

N–Aryl bond formation under copper catalysis has played a pivotal role and has been
extensively used as a key step in the total syntheses of several therapeutic molecules. The …

Naphthalene monoimide (NMI) molecules have recently been discovered to act as a
powerful reductant to trigger strong C–Cl bond cleavage reactions. In this report, we explore …

Alcohols and ethers were identified as sustainable methine sources for synthesizing
quinazolinone and benzimidazole derivatives using a combination of TsOH· H2O/O2 and …