Tetrahydro-γ-carbolines (THγ Cs) constitute one of the most important subtypes of indole
alkaloids. In addition to being substructures of natural products, these structural motifs and …

Heterocycles are generally biologically active compounds and find widespread applications
in medicinal chemistry, agricultural science and the fine chemical industry. For the synthesis …

The stereocontrolled total synthesis of (+)-pleiocarpamine and the total syntheses of (+)-
voacalgine A and (+)-bipleiophylline have been achieved. The scalable and concise 10-step …

Herein, we report an unprecedented skeletal rearrangement reaction of tetrahydro‐β‐
carbolines enabled by copper‐catalyzed single‐electron oxidative oxygenation, in which …

We report a safe and convenient open-flask copper-catalyzed selective oxidation/
functionalization methodology for tetrahydrocarbolines and tetrahydro-β-carbolines that …

Oxidative rearrangement of indoles is an essential transformation that has been widely used
in the synthesis of many pharmaceutical agents and bioactive natural products. Herein, we …

One-electron oxidation (OEO) can deeply change the structure and reactivity of organic
molecules. Rings exist ubiquitously in natural products and pharmaceutical molecules. The …

Covering: since early reports up to the end of 2020 This review presents a complete
coverage of the mavacuranes alkaloids since early reports till date. Mavacuranes alkaloids …

Oxidative reactions provide an effective strategy for phenol transformation via conjugated
addition, C–H functionalization, cyclization reactions, etc. It has enabled broad utilization of …

Efficient access to evodiamine and its analogues is presented via Lewis acid catalysis. In
this reaction, three chemical bonds and two heterocyclic-fused rings are constructed in one …