Diaryl and arylheteroaryl urea derivatives as modulators of the 5-HT2A serotonin receptor useful for the prophylaxis and treatment of disorders related thereto
B Teegarden, H Jayakumar, H Li… - US Patent …, 2016 - Google Patents
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Imidazo [1, 2-a] pyridine derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto
Y Xiong, K Feichtinger, AS Ren, B Ullman - US Patent 9,567,327, 2017 - Google Patents
5,128,351 A 7, 1992 Wissner schizophrenia and related disorders, diabetic-related disor
5,523,280 A 6, 1996 Chene et al. ders, progressive multifocal leukoencephalopathy and the …
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Diaryl and arylheteroaryl urea derivatives as modulators of the 5-HT2A serotonin receptor useful for the prophylaxis and treatment of disorders related thereto
B Teegarden, H Jayakumar, H Li… - US Patent …, 2017 - Google Patents
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Processes for preparing substituted N-aryl-N′-[3-(1H-pyrazol-5-YL) phenyl] ureas and intermediates thereof
JR Fritch, FM Carleton, EA Lally, H Li… - US Patent …, 2010 - Google Patents
(54) PROCESSES FOR PREPARING 6,140,509 A 10/2000 Behan et al. SUBSTITUTED
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6,150,393 A 1 1/2000 Behan et al. N-ARYL-N'-3-(1H-PYRAZOL-5-YL) PHENYL 6,271,261 …
3-Phenyl-pyrazole derivatives as modulators of the 5-HT2a serotonin receptor useful for the treatment of disorders related thereto
B Teegarden, Y Xiong, S Strah-Pleynet… - US Patent …, 2011 - Google Patents
First worldwide family litigation filed litigation Critical https://patents. darts-ip. com/? family=
36218810&utm_source= google_patent&utm_medium= platform_link&utm_campaign …
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Pyrazole derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto
Y Xiong, MC Cherrier, JSK Choi, PI Dosa… - US Patent …, 2016 - Google Patents
(57) ABSTRACT Pyrazole derivatives of Formula (Ia) and pharmaceutical compositions
thereof that modulate the activity of the sero tonin 5HT2 receptor. Formula (Ia). Compounds …
thereof that modulate the activity of the sero tonin 5HT2 receptor. Formula (Ia). Compounds …
Diaryl and arylheteroaryl urea derivatives as modulators of the 5-HT2A serotonin receptor useful for the prophylaxis and treatment of disorders related thereto
B Teegarden, H Jayakumar, H Li… - US Patent …, 2014 - Google Patents
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Ethers, secondary amines and derivatives thereof as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto
B Teegarden, D Chapman, M Decaire, PI Dosa… - US Patent …, 2012 - Google Patents
The present invention pertains to certain compounds of For mula (Ia) and pharmaceutical
compositions thereof that modulate the activity of the 5-HT2A serotonin receptor …
compositions thereof that modulate the activity of the 5-HT2A serotonin receptor …
Primary amines and derivatives thereof as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto
B Teegarden, D Chapman, J Choi… - US Patent …, 2012 - Google Patents
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3-Phenyl-Pyrazole Derivatives as Modulators of the 5-Ht2A Serotonin Receptor Useful for the Treatment of Disorders Related Thereto
B Teegarden, Y Xiong, S Strah-Pleynet… - US Patent App. 11 …, 2007 - Google Patents
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