Synthesis and evaluation of novel xanthene‐based thiazoles as potential antidiabetic agents

S Naseem, Z Shafiq, P Taslimi, S Hussain… - Archiv der …, 2023 - Wiley Online Library
A series of xanthene‐based thiazoles was synthesized and characterized by different
scpectroscopic methods, ie Proton nuclear magnetic resonance (1H NMR), carbon nuclear …

The assembly of integrated continuous flow platform for on-demand rosiglitazone and pioglitazone synthesis

M Purwa, A Rana, AK Singh - Reaction Chemistry & Engineering, 2022 - pubs.rsc.org
Manufacturing thiazolidinediones in a batch process is often carried out at different
locations, where each successive batch collects a certain amount of intermediate followed …

Synthesis of thiazolidin-4-ones and thiazinan-4-ones from 1-(2-aminoethyl) pyrrolidine as acetylcholinesterase inhibitors

AM das Neves, GA Berwaldt, CT Avila… - Journal of Enzyme …, 2020 - Taylor & Francis
The present study describes the synthesis of a novel series of thiazolidin-4-one and
thiazinan-4-one using 1-(2-aminoethyl) pyrrolidine as amine precursor. All compounds were …

Dehydroabietylamine-based thiazolidin-4-ones and 2-thioxoimidazolidin-4-ones as novel tyrosyl-DNA phosphodiesterase 1 inhibitors

K Kovaleva, E Mamontova, O Yarovaya, O Zakharova… - Molecular Diversity, 2021 - Springer
Abstract Tyrosyl-DNA phosphodiesterase 1 (TDP1) is a DNA repair enzyme that plays a key
role in repairing damage caused by various antitumor drugs. It is a promising target in …

Synthesis, identification of some new derivatives of 4-amino antipyrine bearing six and seven membered rings

SA Alsahib, SR Baqer - Journal of Physics: Conference Series, 2021 - iopscience.iop.org
In this paper, we consider the Synthesis of a series of various 4-amino antipyrine derivatives
containing 1, 3-thiazinan-4-one, 1, 3-oxazinan-6-one, and 1, 3-oxazepin-4, 7-dione in its …

Síntese e avaliação do potencial anticolinesterásico de tiazolidin-4-onas tendo como precursor a 2-cicloexilmetilamina

BC Moreira - 2021 - repositorio.ufpel.edu.br
Wilson Cunico. 2021. 989 fls. Dissertação (Mestrado Bioquímica e Bioprospecção)-Centro
de Ciências Químicas, Farmacêuticas e de Alimentos, Universidade Federal de Pelotas …

Síntese e Avaliação In Vitro da Atividade Antiglioma, Antioxidante e Inibidora da Monoaminoxidase-B de 2-imino-tiazolidin-4-onas

JCC Júnior - 2020 - repositorio.ufpel.edu.br
A series of novel 2-imino-4-thiazolidinone (5a-p) derivatives was synthesized and evaluated
for their cytotoxic activity against glioma (C6) cancer cell line, on the other hand, this work …

[PDF][PDF] Kseniya Kovaleva, Evgeniya Mamontova, Olga Yarovaya, Olga Zakharova, Alexandra Zakharenko, Olga Lavrik &

N Salakhutdinov - researchgate.net
Abstract Tyrosyl-DNA phosphodiesterase 1 (TDP1) is a DNA repair enzyme that plays a key
role in repairing damage caused by various antitumor drugs. It is a promising target in …

Suplementação de butirato para prevenção de diarreia e no desenvolvimento gastrointestinal e corporal de bezerros leiteiros

MG Victor - 2020 - repositorio.ufpel.edu.br
Resumo VICTOR, Melinda Gomes. 3, 5-Di-terc-butil-4-hidroxibenzaldeído como precursor
para a síntese de novas 1, 3-tiazolidin-4-onas e potencial antioxidante via captura de …