[PDF][PDF] The antioxidant activity of some acylhydrazones with dibenzo [a, d][7] annulene moiety

LI Socea, DC Visan, SF Barbuceanu… - Rev Chim …, 2018 - researchgate.net
Searching new antioxidants compounds to prevent or reduce the impact of oxidative stress
on cells, we designed and synthesized several N-acylhydrazone derivatives with dibenzo [a …

In-silico Molecular Docking and ADMET predictions of Pyrido[2,3-d]pyrimidine-2,4(1H,3H)-Dione Analogues as promising Antimicrobial, Antioxidant and Anticancer …

M Sivanandhan, A Parasuraman - Polycyclic Aromatic Compounds, 2024 - Taylor & Francis
Pyridopyrimidine are heterocyclic molecules enclosing fused pyridine and pyrimidine rings.
Owing to its fascinating core structure and pharmacological applications a series of 7-([1 …

A novel bidentate ligand containing oxime, hydrazone and indole moieties and its BF2+ bridged transition metal complexes and their efficiency against prostate and …

I Babahan, A Özmen, M Aksel, MD Bilgin… - Applied …, 2020 - Wiley Online Library
In this study, a novel bidentate ligand containing oxime, hydrazone, and indole moieties and
its BF2+‐bridged transition metal complexes [Ni (II), Cu (II), and Co (II)] were synthesized …

QSAR classification model for diverse series of antifungal agents based on improved binary differential search algorithm

AM Al-Fakih, ZY Algamal, MH Lee, M Aziz… - SAR and QSAR in …, 2019 - Taylor & Francis
An improved binary differential search (improved BDS) algorithm is proposed for QSAR
classification of diverse series of antimicrobial compounds against Candida albicans …

[PDF][PDF] Synthesis of azolines and imidazoles and their use in drug design

A Reyes-Arellano, O Gómez-García… - Med Chem (Los …, 2016 - academia.edu
Heterocycles are very important functional groups, especially in medicinal chemistry. They
are not only pivotal in the synthesis of drugs, but also form part of the structure of a diversity …

Quantitative structure-activity relationship model for classifying the diverse series of antifungal agents using ratio weighted penalized logistic regression

AM Alharthi, MH Lee, ZY Algamal… - SAR and QSAR in …, 2020 - Taylor & Francis
One of the most challenging issues when facing a Quantitative structure-activity relationship
(QSAR) classification model is to deal with the descriptor selection. Penalized methods have …

Electrochemical-Promoted Synthesis of 2-Thiazolines via Selenylation/Cyclization of N-Allylthioamides

C Pan, P Liu, A Wu, M Li, L Wen… - Chinese Journal of Organic …, 2020 - sioc-journal.cn
An electrochemical selenylation/cyclization of N-allylthioamides has been developed for the
synthesis of selenium-containing 2-thiazolines. This protocol provides an efficient approach …

New pyrimidines and triazolopyrimidines as antiproliferative and antioxidants with cyclooxygenase-1/2 inhibitory potential

AM Omar, HA Abd El Razik, AA Hazzaa… - Future Medicinal …, 2019 - Taylor & Francis
Aim: Cyclooxygenase-2 (COX-2) inhibition and scavenging-free radicals are important
targets in cancer treatment. Materials & methods: Sulfanylpyrimidines and …

A series of furan-based hydrazones: design, synthesis, and evaluation of antimicrobial activity, cytotoxicity and genotoxicity

MD Altintop, B Sever, ÖA Eklioğlu… - Letters in Drug …, 2020 - ingentaconnect.com
Background: Hydrazones, frequently occurring motifs in many bioactive molecules, have
attracted a great deal of interest as potent antimicrobial agents. Objective: The aim of this …

Two Neglected multicomponent reactions: Asinger and Groebke reaction for constructing thiazolines and imidazolines

ZQ Liu - Current Organic Synthesis, 2015 - ingentaconnect.com
The multicomponent reaction (MCR) is an important research field in the organic synthetic
methodology. In 1956, Professor Friedrich Asinger reported a method for synthesizing …