Asymmetric Synthesis and Biological Evaluation of Platensilin, Platensimycin, Platencin, and Their Analogs via a Bioinspired Skeletal Reconstruction Approach

ZX Gao, H Wang, AH Su, QY Li, Z Liang… - Journal of the …, 2024 - ACS Publications
Platensilin, platensimycin, and platencin are potent inhibitors of β-ketoacyl–acyl carrier
protein synthase (FabF) in the bacterial and mammalian fatty acid synthesis system …