Abstract Initially, the Atherton–Todd (AT) reaction was applied for the synthesis of
phosphoramidates by reacting dialkyl phosphite with a primary amine in the presence of …

Our previous work demonstrated that Wnt16 expression in cisplatin-damaged tumor-
associated fibroblasts is a key factor contributing to cisplatin resistance in malignancies …

There remain gaps in our understanding of the fate of liposomes in the infant gastrointestinal
tract, especially regarding essential proteins such as lactoferrin. Models in vitro that mirrored …

In this study, the concept of dynamic combinatorial chemistry (DCC) was applied to explore
novel cholesterol esterase (CEase) inhibitors. In the presence of enzyme, two substrates …

The instability of liposomal delivery system during passaging through the gastrointestinal
tract (GIT) stimulates a demand to find a stable liposome. This research studied the …

We present a new class of inhibitors of pancreatic cholesterol esterase (CEase) based on
'priviledged'5-benzylidenerhodanine and 5-benzylidene-2, 4-thiazolidinedione structural …

A series of phosphorylated flavonoids were synthesized and investigated in vitro as
inhibitors of pancreatic cholesterol esterase (CEase) and acetylcholinesterase (AChE). The …

以功能因子对α-淀粉酶, α-葡萄糖苷酶, 胰脂肪酶, 胆固醇酯酶和胆固醇胶束溶解度抑制率为评价
指标, 筛选出5 种活性成分. 以α-淀粉酶和胆固醇酯酶活性为评价指标, 用正交t …

This study investigated the hypocholesterolaemic effects of bitter melon aqueous extracts
(BMAE) in vitro, the inhibitory effects of BMAE on pancreatic cholesterol esterase (CEase) …

Nutraceuticals are defined as a food or food ingredients that prevent and treat diseases.
They contain dietary supplements like proteins, vitamins and minerals, compound derived …