[HTML][HTML] Antimicrobial activity of 1, 3, 4-oxadiazole derivatives

T Glomb, P Świątek - International journal of molecular sciences, 2021 - mdpi.com
The worldwide development of antimicrobial resistance forces scientists to search for new
compounds to which microbes would be sensitive. Many new structures contain the 1, 3, 4 …

[HTML][HTML] Synthetic approaches and pharmacological activity of 1, 3, 4-oxadiazoles: a review of the literature from 2000–2012

CS De Oliveira, BF Lira, JM Barbosa-Filho… - Molecules, 2012 - mdpi.com
Molecules | Free Full-Text | Synthetic Approaches and Pharmacological Activity of 1,3,4-Oxadiazoles:
A Review of the Literature from 2000–2012 Next Article in Journal Chemical Composition of …

Design, synthesis, and evaluation of new sulfone derivatives containing a 1, 3, 4-oxadiazole moiety as active antibacterial agents

P Li, D Hu, D Xie, J Chen, L Jin… - Journal of agricultural and …, 2018 - ACS Publications
This study aimed to synthesize some new sulfone derivatives containing a 1, 3, 4-oxadiazole
moiety and investigate their in vitro antibacterial activities against Xanthomonas oryzae pv …

Synthesis and antifungal activity of 3-(1, 3, 4-oxadiazol-5-yl)-indoles and 3-(1, 3, 4-oxadiazol-5-yl) methyl-indoles

MZ Zhang, N Mulholland, D Beattie, D Irwin… - European Journal of …, 2013 - Elsevier
On the basis of the principle of combination of active structural moieties, a modified and
efficient synthetic method for three series of novel indole-based 1, 3, 4-oxadiazoles is …

Design, synthesis, characterization, molecular docking studies and anticancer activity evaluation of novel hydrazinecarbothioamide, 1, 2, 4-triazole-3-thione, 4 …

ED Dincel, Ç Akdağ, T Kayra, ED Coşar… - Journal of Molecular …, 2022 - Elsevier
A series of novel hydrazinecarbothioamide, 1, 2, 4-triazole-3-thione, 4-thiazolidinone and 1,
3, 4-oxadiazole derivatives were synthesized and evaluated for their cytotoxic activity …

Novel bisthioether derivatives containing a 1, 3, 4‐oxadiazole moiety: design, synthesis, antibacterial and nematocidal activities

P Li, P Tian, Y Chen, X Song, W Xue… - Pest management …, 2018 - Wiley Online Library
BACKGROUND The literature shows that bisthioether and 1, 3, 4‐oxadiazole derivatives
exhibit a wide variety of biological activities. In this study, a series of novel bisthioether …

Review of synthesis of 1, 3, 4-oxadiazole derivatives

KD Patel, SM Prajapati, SN Panchal… - Synthetic …, 2014 - Taylor & Francis
Oxadiazole nucleus shows a broad spectrum of pharmaceutical applications. Thus, in recent
years scientists have developed various new methods for the synthesis of its derivatives …

Design, synthesis, and antibacterial activity against rice bacterial leaf blight and leaf streak of 2, 5-substituted-1, 3, 4-oxadiazole/thiadiazole sulfone derivative

P Li, L Shi, X Yang, L Yang, XW Chen, F Wu… - Bioorganic & medicinal …, 2014 - Elsevier
Abstract A series of 2, 5-substituted-1, 3, 4-oxadiazole/thiadiazole sulfone derivatives were
synthesized and evaluated for their antibacterial activities against rice bacterial leaf blight …

Synthesis and Bioactivity Evaluation of Novel Arylimines Containing a 3-Aminoethyl-2-[(p-trifluoromethoxy)anilino]-4(3H)-quinazolinone Moiety

X Wang, P Li, Z Li, J Yin, M He, W Xue… - Journal of agricultural …, 2013 - ACS Publications
Twenty-seven novel (E)-3-[2-arylideneaminoethyl]-2-[4-(trifluoromethoxy) anilino]-4 (3 H)-
quinazolinone derivatives were synthesized by reacting various aromatic aldehydes with …

New oxadiazoles with selective-COX-2 and EGFR dual inhibitory activity: Design, synthesis, cytotoxicity evaluation and in silico studies

NA El-Sayed, MS Nour, MA Salem, RK Arafa - European Journal of …, 2019 - Elsevier
Novel heterocyclic oxadiazoles viz. 2-subsituted-5-(4-pyridyl)-1, 3, 4-oxadiazoles, 2-
subsituted-5-(3-pyridyl)-1, 3, 4-oxadiazoles and 2-subsituted-5-(phenyl or 4-chlorophenyl-1 …