Androgen receptor heterogeneity and phosphorylation in human LNCaP cells
JH Van Laar, J Bolt-de Vries, ND Zegers… - Biochemical and …, 1990 - Elsevier
Androgen receptor heterogeneity and phosphorylation were studied in the human LNCaP
cell line. Fluorography after photoafffinity labeling as well as immunoblotting with a specific …
cell line. Fluorography after photoafffinity labeling as well as immunoblotting with a specific …
Steroid hormone receptors
EV Jensen - Cell Receptors: Morphological Characterization and …, 1991 - Springer
The steroid hormones comprise a large and important family of cell regulators. These
include sex hormones (estrogens, progestins, androgens), adrenal cortical hormones …
include sex hormones (estrogens, progestins, androgens), adrenal cortical hormones …
Antiestrogenic activity of two 11β-estradiol derivatives on MCF-7 breast cancer cells
L Jin, M Borrás, M Lacroix, N Legros, G Leclercq - Steroids, 1995 - Elsevier
Two 11β-derivatives of estradiol (E2) were tested for their potential antiestrogenic activity in
the MCF-7 breast cancer model: one contained a phenoxydimethylaminoethyl side-chain …
the MCF-7 breast cancer model: one contained a phenoxydimethylaminoethyl side-chain …
In vitro phosphorylation and hormone binding activation of the synthetic wild type human estradiol receptor
A Migliaccio, G Castoria, A de Falco… - The Journal of Steroid …, 1991 - Elsevier
A tyrosine kinase purified from calf uterus activates the hormone binding of endogenous
estradiol receptor (ER) predephosphorylated and preinactivated by a nuclear …
estradiol receptor (ER) predephosphorylated and preinactivated by a nuclear …
Estrogen effects in the heart
T Pelzer, A Shamim, L Neyses - Biochemical Mechanisms in Heart …, 1996 - Springer
Gender specific differences in cardiovascular disease are largely mediated by sex
hormones. The use of estrogens significantly reduces the overall incidence of heart disease …
hormones. The use of estrogens significantly reduces the overall incidence of heart disease …
The role of estradiol receptor in the proliferative activity of vanadate on MCF-7 cells
Vanadate stimulates growth of the estradiol-responsive MCF-7 cells in the absence of
estrogens through a mechanism requiring tyrosine kinase activity. The proliferative effect of …
estrogens through a mechanism requiring tyrosine kinase activity. The proliferative effect of …
Identification of a novel phosphorylation site in human androgen receptor by mass spectrometry
Z Zhu, RR Becklin, DM Desiderio, JT Dalton - Biochemical and Biophysical …, 2001 - Elsevier
An N-terminal hexahistidine-tagged full-length human androgen receptor protein (His6-hAR)
was overexpressed and purified to apparent homogeneity in the presence of …
was overexpressed and purified to apparent homogeneity in the presence of …
Threonine on amino acid position 868 in the human androgen receptor is essential for androgen binding specificity and functional activity
C Risstalpers, MCT Verleunmooijman… - Biochemical and …, 1993 - Elsevier
The human androgen receptor gene in the androgen sensitive prostate tumor cell line
(LNCaP) contains a point mutation in codon 868 resulting in the substitution of threonine by …
(LNCaP) contains a point mutation in codon 868 resulting in the substitution of threonine by …
Cloning and sequencing of the gilthead sea bream estrogen receptor cDNA
JA Munoz-Cueto, E Burzawa-Gérard, O Kah… - DNA …, 1999 - Taylor & Francis
We report here the complete nucleotide sequence of a cDNA clone containing the full-
coding sequence of the Sparus aurata estrogen receptor (ER) isolated from an expression …
coding sequence of the Sparus aurata estrogen receptor (ER) isolated from an expression …
Modulators of cellular protein phosphorylation alter thetrans-activation function of human progesterone receptor and the biological activity of progesterone …
DP Edwards, NL Weigel, SK Nordeen… - Breast cancer research …, 1993 - Springer
Addition of progesterone to breast cancer cells in vivo increases phosphorylation of human
progesterone receptor (PR), suggesting that phosphorylation has a regulatory role in …
progesterone receptor (PR), suggesting that phosphorylation has a regulatory role in …