Tetrahydroquinoline is one of the most important simple nitrogen heterocycles, being
widespread in nature and present in a broad variety of pharmacologically active …

A review of the recent literature is given focusing on synthetic approaches to 1, 2, 3, 4-
tetrahydroquinolines, 2, 3-dihydro-4 (1 H)-quinolinones and 4 (1 H)-quinolinones using …

The AT-rich mitochondrial DNA (kDNA) of trypanosomatid parasites is a target of DNA minor
groove binders. We report the synthesis, antiprotozoal screening, and SAR studies of three …

We report herein a mild stereo‐and regioselective dearomatization of quinolines using the
simple low valent HCo (N2)(PPh3) 3 complex that exhibits labile ligands. Conditions to form …

A highly selective and divergent synthesis which enabled access to various complex
compounds is highly attractive in organic synthesis and medicinal chemistry. Herein, we …

The enantioselective Povarov reaction is one of the most powerful synthetic strategy to
synthesize chiral, highly functionalized 1, 2, 3, 4‐tetrahydroquinolines. The present …

Herein, we report the preparation of a panel of Schiff bases analogues as antiprotozoal
agents by modification of the stereoelectronic effects of the substituents on N-1 and N-4 and …

We report an efficient use of bimetallic PdRh alloy nanoparticles on Fe 3 O 4 for
chemoselective quinoline hydrogenation to 1, 2, 3, 4-tetrahydroquinoline with ammonia …

This article describes the characterization of various encapsulated formulations of
benznidazole, the current first-line drug for the treatment of Chagas disease. Given the …

An asymmetric enantioselective flow process is reported for the formal synthesis of a 1, 2, 3,
4‐tetrahydroquinoline selective estrogen receptor modulator. Starting from an easily …