Cytostatic tetrazole–butenolide conjugates: linking tetrazole and butenolide rings via stille coupling and biological activity of the target substances

V Balšánek, L Tichotova, J Kuneš… - Collection of …, 2009 - cccc.uochb.cas.cz
A series of tetrazoles linked to the butenolide core via benzene rings were prepared by the
Stille coupling reaction of α-(tributylstannyl) butenolides and 5-(alkylsulfanyl)-1-(4 …

Metabolic profiling of a potential antifungal drug, 3-(4-bromophenyl)-5-acetoxymethyl-2, 5-dihydrofuran-2-one, in mouse urine using high-performance liquid …

M Nobilis, M Pour, P Šenel, J Pavlík, J Kuneš… - … of Chromatography B, 2007 - Elsevier
3-(4-Bromophenyl)-5-acetyloxymethyl-2, 5-dihydrofuran-2-one (LNO-18-22) is a
representative member of a novel group of potential antifungal drugs, derived from a natural …

Synthesis and anti-fungal properties of some simple cyclopentenones and derivatives

JA Miller, AW Pugh, GM Ullah, GM Welsh - Tetrahedron Letters, 2001 - Elsevier
1-Methylsulphenyl-2-phenylsulphenylethyne has been shown to be a precursor for either α-
sulphenyl ketone or α-methylene ketone moieties in cyclopentenoids produced via [3+ 2] …

Pentenolide Analogues of Antifungal Butenolides: Strategies Towards 3, 6-Disubstituted Pyranones and Unexpected Loss of Biological Effect

I Šnajdr, J Pavlik, R Schiller, J Kuneš… - Collection of …, 2007 - cccc.uochb.cas.cz
Pentenolide analogues of antifungal 3, 5-disubstituted butenolides were prepared by
oxidative cyclization of 2-(substituted aryl) hex-5-enoic acids as the key step. Given the …

A Concise Synthesis of (−)‐Incrustoporin and its Analogues by Pd–catalyzed Suzuki‐Miyaura Coupling from γ‐Vinyl‐γ‐butyrolactone

JL Nallasivam, RA Fernandes - ChemistrySelect, 2016 - Wiley Online Library
A highly efficient synthesis of C3‐arylbutenolides by Suzuki‐Miyaura coupling is described.
We developed a simple protocol to accomplish scaffolds of C3‐arylbutenolides which …

Ultrasound-Mediated Willgerodt–Kindler Reactions: Non-thermal Synthesis of Thioacetamides

MM Mojtahedi, T Alishiri, MS Abaee - Phosphorus, Sulfur, and …, 2011 - Taylor & Francis
Non-thermal, solvent-free condensation of several aryl methyl ketones with amines and
elemental sulfur is efficiently conducted using ultrasonic irradiation within short time periods …

Synthesis and herbicidal activities of 1, 3, 4-thiadiazole derivatives of 5-(fluoro-substituted phenyl)-2-furamide

WD Bian, A Chai, SR Yu, SJ Xue - Chinese Journal of Organic …, 2008 - sioc-journal.cn
Abstract Twenty new N-(5-aryl-1, 3, 4-thiadiazol-2-yl)-5-(fluorophenyl)-2-furamides were
designed, and characterized by elemental analysis, IR and 1H NMR spectra. The …

Progress in the Formation of Carbon-Hetero Bond Based on 2 (5H)-Furanones

YH TAN, JX LI, WK HONG, CY WANG - Chinese Journal of Organic …, 2011 - sioc-journal.cn
Recently, the organic synthesis based on 2 (5H)-furanones (1) has attracted much attention
owing to the unique carbon skeleton of 2 (5H)-furanone which is widely present in a variety …

Synthesis and Biological Activities of Vicinal Diaryl Furans

NR Patel, DV Patel - Vicinal Diaryl Substituted Heterocycles, 2018 - Elsevier
Furans are considered an influential part of heterocyclic systems due to their interesting
biological properties. Vicinal diaryl furans have shown significant biological activities such …

[引用][C] 微波诱导合成5-芳氧亚甲基-2-[5′-(4 ″-氯代苯基)-2′-呋喃甲酰胺基]-1, 3, 4-噁二唑

杨靖亚, 王俊科, 李政, 王喜存 - 西北师范大学学报: 自然科学版, 2003