[HTML][HTML] Functional Pyrazolo[1,5-a]pyrimidines: Current Approaches in Synthetic Transformations and Uses As an Antitumor Scaffold

A Arias-Gomez, A Godoy, J Portilla - Molecules, 2021 - mdpi.com
Pyrazolo [1, 5-a] pyrimidine (PP) derivatives are an enormous family of N-heterocyclic
compounds that possess a high impact in medicinal chemistry and have attracted a great …

Modern Trends of Organic Chemistry in Russian Universities

AI Konovalov, IS Antipin, VA Burilov… - Russian Journal of …, 2018 - Springer
This review is devoted to the scientific achievements of the departments of organic chemistry
in higher schools of Russia within the past decade.

5-Amino-pyrazoles: potent reagents in organic and medicinal synthesis

A Shaabani, MT Nazeri, R Afshari - Molecular diversity, 2019 - Springer
Amino-pyrazoles have proven to be a class of fascinating and privileged organic tools for the
construction of diverse heterocyclic or fused heterocyclic scaffolds. This review presents …

Integrated pyrazolo [1, 5-a] pyrimidine–hemicyanine system as a colorimetric and fluorometric chemosensor for cyanide recognition in water

A Tigreros, HA Rosero, JC Castillo, J Portilla - Talanta, 2019 - Elsevier
A new probe for cyanide detection based on the integrated pyrazolo [1, 5-a] pyrimidine–
hemicyanine (PpHe) system was synthesized in an efficient and straightforward manner …

[PDF][PDF] Recent advances in the synthesis of new pyrazole derivatives

JC Castillo, J Portilla - Targets Heterocycl. Syst, 2018 - soc.chim.it
Pyrazoles have attracted great attention in organic and medicinal chemistry, due to their
proven utility as synthetic intermediates for the preparation of diverse bioactive compounds …

Simple access toward 3-halo-and 3-nitro-pyrazolo [1, 5-a] pyrimidines through a one-pot sequence

JC Castillo, HA Rosero, J Portilla - RSC advances, 2017 - pubs.rsc.org
Herein, a regioselective, time-efficient and one-pot route for the synthesis of diversely
substituted 3-halo-and 3-nitropyrazolo [1, 5-a] pyrimidines in good to excellent yields …

[PDF][PDF] Современные тенденции органической химии в университетах России

АИ Коновалов, ИС Антипин, ВА Бурилов… - Журнал …, 2018 - researchgate.net
5. Кафедра органической химии Московского государственного университета им. МВ
Ломоносова. 6. Кафедра химии Российского национального исследовательского …

Lewis‐acid Promoted Chemoselective Condensation of 2‐Aminobenzimidazoles or 3‐Aminoindazoles with 3‐Ethoxycyclobutanones to Construct Fused Nitrogen …

W Kong, Y Zhou, Q Song - Advanced Synthesis & Catalysis, 2018 - Wiley Online Library
A Lewis‐acid promoted chemoselective condensation of 2‐aminobenzimidazoles or 3‐
aminoindazoles with 3‐ethoxycyclobutanones is presented. Diverse fused heterocycles …

Conjugated enynones: Preparation, properties and applications in organic synthesis

AA Golovanov, IS Odin, SS Zlotskii - Russian Chemical Reviews, 2019 - iopscience.iop.org
Published data on the preparation methods, properties and chemical transformations of
linear-and cross-conjugated enynones are integrated. The molecular and crystal structures …

Reactivity of cross-conjugated enynones in cyclocondensations with hydrazines: Synthesis of pyrazoles and pyrazolines

AA Golovanov, IS Odin, DM Gusev… - The Journal of …, 2021 - ACS Publications
The cyclocondensation of cross-conjugated enynones, dienynones, and trienynones (easily
available due to low-cost starting compounds) with arylhydrazines leads to the …