Heterocyclic compounds are a class of compounds that is deeply intertwined with biological
processes and is found in about 90% of commercially available medicines. They serve a …

An efficient copper–iodine co-catalyzed 2, 3-difunctionalization of indoles with azoles and
phenols via temperature-controlled selectivity switch has been developed for the green …

The combination of organolithium chemistry with gold catalysis has enabled the
development of a synthetic strategy for accessing polysubstituted indoles and carbazoles …

A p-toluenesulfonic acid-catalyzed cascade reaction is reported for the synthesis of 4-
functionalized tetrahydrocarbazolones via the reaction of 4-(indol-2-yl)-4-oxobutanal …

Indoles are extremely important and versatile building blocks in the field of chemistry. This
review highlights the advance made in the three‐component reactions of indoles between …

A synthetic strategy for the construction of 2, 2‐disubstituted indolin‐3‐ones from 2‐
alkynylnitroarenes and ketones has been described. The corresponding indolin‐3‐one …

The Ritter-type reaction, without relying on a pre-installed functional group, is a highly
efficient tool for the construction of amides. However, the intrinsic chemo-selectivity that …

Herein we present a transition-metal-free cross-coupling reaction of isatogens with boronic
acids through a 1, 4-metalate shift of a boron “ate” complex. This coupling reaction provides …

A highly efficient oxidative dearomatization of indoles with H-phosphorus oxides in the
presence of TEMPO oxoammonium salt has been demonstrated. Through the intramolecular …

We have explored a one-pot, tandem protocol for constructing a linear tetracyclic aromatic
core isoindoloindolone via FeCl 3-mediated annulative coupling of 2-aminoacetophenones …