Synthesis of 9-Cinnamyl-9H-purine Derivatives as Novel TLR4/MyD88/NF-κB Pathway Inhibitors for Anti-inflammatory Effects

L Pham, R Jiang, Z Liu, M Nguyen… - ACS Medicinal …, 2023 - ACS Publications
The novel 9-cinnamyl-9 H-purine skeleton, inspired by resveratrol and curcumin, was
developed to avoid a pan-assay interference compound (PAINS) related to invalid metabolic …