Melatonin has a key role in the circadian rhythm relay to periphery organs. Melatonin exerts
its multiple roles mainly through two seven transmembrane domain, G-coupled receptors …

Publications from both academic and industry on the synthesis and application of chemical
libraries continued at a rapid pace in 2000. The total number of libraries cited was 284 …

A novel series of melatonin receptor ligands, characterized by a N-(substituted-anilinoethyl)
amido scaffold, along with preliminary structure–activity relationships (SARs), is presented …

The amination of racemic α‐chiral aldehydes, 2‐phenylpropanal derivatives, was
investigated employing ω‐transaminases. By medium and substrate engineering the optical …

Conformationally restricted phenalene and acenaphthene derivatives 5 were synthesized
from phenalen-1-one and acenaphthen-1-one derivatives using the Horner− Emmons …

A series of phenoxyalkyl and phenylthioalkyl amides were prepared as melatoninergic
ligands. Modulation of affinity of the newly synthesized compound by applying SARs around …

A series of substituted N-[3-(3-methoxyphenyl) propyl] amides were synthesized and their
binding affinities towards human melatonin MT1 and MT2 receptors were evaluated. It was …

A novel series of melatonin receptor ligands was discovered by opening the cyclic scaffolds
of known classes of high affinity melatonin receptor antagonists, while retaining the …

Amido derivatives 10–18 of the corresponding oxyamines were synthesised as
melatoninergic ligands by the reaction of hydroxyphtalimide with the halogeno derivatives or …

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