[HTML][HTML] An overview on the antibacterial properties of juglone, naphthazarin, plumbagin and lawsone derivatives and their metal complexes
C Majdi, V Duvauchelle, P Meffre… - Biomedicine & …, 2023 - Elsevier
Bacterial resistance development represents a serious threat to human health across the
globe and has become a very serious clinical problem for many classes of antibiotics …
globe and has become a very serious clinical problem for many classes of antibiotics …
Design, synthesis, spectroscopic characterization, single crystal X-ray analysis, in vitro α-amylase inhibition assay, DPPH free radical evaluation and computational …
In our quest to design and develop N/O-containing inhibitors of α-amylase, we have tried to
synergize the inhibitory action of 1, 4-naphthoquinone, imidazole and 1, 2, 3-triazole motifs …
synergize the inhibitory action of 1, 4-naphthoquinone, imidazole and 1, 2, 3-triazole motifs …
New naphthoquinone thiazole hybrids as carbonic anhydrase and cholinesterase inhibitors: Synthesis, crystal structure, molecular docking, and acid dissociation …
Abstract In this study, N-[3-(3-amino-1, 4-dioxo-1, 4-dihydronaphthalen-2-yl)-4-R-thiazol-2
(3H)-ylidene]-2, 6-difluorobenzamide derivatives as new 1, 4-naphthoquinone thiazole …
(3H)-ylidene]-2, 6-difluorobenzamide derivatives as new 1, 4-naphthoquinone thiazole …
Anti‐inflammatory Potential of 1, 4‐Naphthoquinone Acyl Thiourea Hybrids on Lipopolysaccharide‐Activated Mammalian Macrophages, and Their Acid Dissociation …
In this study, seven new and known 1, 4‐naphthoquinone acyl thiourea hybrids were
synthesized and their molecular structures were confirmed by various analytical methods …
synthesized and their molecular structures were confirmed by various analytical methods …
[HTML][HTML] Hybrids of 1, 4-Naphthoquinone with Thymidine Derivatives: Synthesis, Anticancer Activity, and Molecular Docking Study
M Kadela-Tomanek, K Krzykawski, A Halama… - Molecules, 2023 - mdpi.com
One of the most essential health problems is cancer, the first or second cause of death
worldwide. Head and neck cancers are hard to detect due to non-specific symptoms. The …
worldwide. Head and neck cancers are hard to detect due to non-specific symptoms. The …
Synthesis of water-soluble novel bioactive pyridine-based azo coumarin derivative and competitive cytotoxicity, DNA binding, BSA binding study, and in silico analysis …
The diazo coupliling reaction of 3-amino pyridine with coumarin in water medium produces
water soluble 6-[3-pyridyl] azocoumarin. The synthesised compound has been fully …
water soluble 6-[3-pyridyl] azocoumarin. The synthesised compound has been fully …
[HTML][HTML] KuQuinones: a ten years tale of the new pentacyclic quinoid compound
Quinones are widespread in nature, as they participate, mainly as redox mediators, in
several biochemical processes. Up to now, various synthetic quinones have been …
several biochemical processes. Up to now, various synthetic quinones have been …
Design, synthesis, and evaluation of 1, 4-naphthoquinone-chromene hybrids as potential anti-K562 and A549 agents
WH Zhang, B Zhang, BW Pan, XW Liu, ZG Yin… - New Journal of …, 2024 - pubs.rsc.org
Two series of 1, 4-naphthoquinone-chromone hybrids 4a (4aa–4ao) and 4b (4ba–4bq) were
designed, synthesized and evaluated as antitumor agents. Most of the compounds exhibited …
designed, synthesized and evaluated as antitumor agents. Most of the compounds exhibited …
Novel chalcone scaffolds of benzothiophene as an efficient real time hydrazine sensor: Synthesis and single crystal XRD studies
Continue to our on-going research, this article demonstrate the design and development of
an efficient real time hydrazine sensor. A series of novel chalcone scaffolds are synthesised …
an efficient real time hydrazine sensor. A series of novel chalcone scaffolds are synthesised …
Synthesis, Enzyme Inhibition, and Acid Dissociation Constant of 1, 4-Naphthoquinone Thiazole Hybrid
Y Nural, Y Demir - Hacettepe University Journal of the Faculty of …, 2024 - dergipark.org.tr
Bu çalışmada, yeni naftokinon tiyazol hibriti 3 1-((3r, 5r, 7r)-adamantan-1-il)-2-bromoetan-1-
on ile naftokinon açil tiyoüre bileşiğinin 2 tepkimesi ile 74% verimle sentezlendi ve …
on ile naftokinon açil tiyoüre bileşiğinin 2 tepkimesi ile 74% verimle sentezlendi ve …