Catalyst‐ and Solvent‐Free Synthesis of N‐Acylhydrazones via Solid‐State Melt Reaction
P Mayurachayakul, N Niamnont… - Asian Journal of …, 2022 - Wiley Online Library
We describe a fast, simple, and effective synthesis of N‐acylhydrazones via a solid‐state
melt reaction under catalyst‐and solvent‐free conditions. The reactions of 2‐furoic …
melt reaction under catalyst‐and solvent‐free conditions. The reactions of 2‐furoic …
Synthesis of Flurbiprofen Based Amide Derivatives as Potential Leads for Diabetic Management: In Vitro α‐glucosidase Inhibition, Molecular Docking and DFT …
This research is based on the synthesis, characterization and in vitro α‐glucosidase
inhibitory activity of fourteen amides (2 a–2 n) of flurbiprofen drug. Seven compounds in the …
inhibitory activity of fourteen amides (2 a–2 n) of flurbiprofen drug. Seven compounds in the …
[PDF][PDF] Synthesis and anti-inflammatory activity of hydrazide-hydrazones bearing anacardic acid and 1, 2, 3-triazole ring based hybrids
A Reddy, NE Kathale - Orient. J. Chem, 2017 - pdfs.semanticscholar.org
ABSTRACT A novel series of hydrazide-hydrazone derivatives 39-50, linked with anacardic
acid motif and 1, 2, 3-triazole ring were synthesized by reacting 4-(1-(2-methoxy-6 …
acid motif and 1, 2, 3-triazole ring were synthesized by reacting 4-(1-(2-methoxy-6 …
Synthesis, Characterization,'ADMET-SAR'Prediction, DPPH Assay, and Anti-Mycobacterium Study of 4-[(substituted benzyl) amino] benzo hydrazides and its …
Background: Hydrazide-hydrazone derivatives have shown diverse biological activities,
such as antitubercular (anti-TB), antibacterial, antifungal, anticancer, anti-inflammatory …
such as antitubercular (anti-TB), antibacterial, antifungal, anticancer, anti-inflammatory …
Synthesis and in vitro evaluation of some hydrazone derivatives as potential antibacterial agents
Z Asim Kaplancikli, M Dilek Altintop… - Letters in Drug …, 2014 - ingentaconnect.com
Nineteen N'-(benzylidene)-2-[(pyrimidin-2-yl) thio] acetohydrazides were obtained via the
nucleophilic addition-elimination reaction of 2-[(pyrimidin-2-yl) thio)] acetohydrazide with …
nucleophilic addition-elimination reaction of 2-[(pyrimidin-2-yl) thio)] acetohydrazide with …
3-Aminothiophene-2-acylhydrazones: Non-toxic, analgesic and anti-inflammatory lead-candidates
Different chemotypes are described as anti-inflammatory. Among them the N-
acylhydrazones (NAH) are highlighted by their privileged structure nature, being present in …
acylhydrazones (NAH) are highlighted by their privileged structure nature, being present in …
[PDF][PDF] Synthesis and crystal structures of benzohydroxamate-coordinated vanadium (V) oxo complexes with aroylhydrazone ligands
SS Qian, X Zhao, J Wang, Z You - Acta Chimica Slovenica, 2015 - pdfs.semanticscholar.org
Abstract Reaction of [VO (acac) 2](where acac= acetylacetonate), benzohydroxamic acid
(Hbha), and two similar aroylhydrazone ligands in methanol produced two …
(Hbha), and two similar aroylhydrazone ligands in methanol produced two …
New hydrazone derivatives of pyrazole-4-carboxaldehydes exhibited anti-inflammatory properties
M Song, B Liu, S Yu, S He, Y Liang, S Li… - Letters in Drug …, 2020 - ingentaconnect.com
Background: Several series of hydrazone derivatives of pyrazole-4-carboxaldehydes (4-11)
were designed and synthesized to screen their inflammatory activity. Methods: The products …
were designed and synthesized to screen their inflammatory activity. Methods: The products …
Discovery of small molecule COX-1 and Akt inhibitors as anti-NSCLC agents endowed with anti-inflammatory action
MD Altıntop, G Akalın Çiftçi, N Yılmaz Savaş… - International Journal of …, 2023 - mdpi.com
Targeted therapies have come into prominence in the ongoing battle against non-small cell
lung cancer (NSCLC) because of the shortcomings of traditional chemotherapy. In this …
lung cancer (NSCLC) because of the shortcomings of traditional chemotherapy. In this …
Antifungal, mosquito deterrent, and larvicidal activity of N-(benzylidene)-3-cyclohexylpropionic acid hydrazide derivatives
Hydrazone derivatives possess good antifungal and insecticidal activities and their
structures are used in pesticide design. In the present study, for the first time, ten hydrazone …
structures are used in pesticide design. In the present study, for the first time, ten hydrazone …