Novel Pyridyl–Oxazole Carboxamides: Toxicity Assay Determination in Fungi and Zebrafish Embryos

S Chen, DL Zhang, CL Ren, WQ Zou, XY Tian, XH Du… - Molecules, 2021 - mdpi.com
Eight novel pyridyl–oxazole carboxamides were evaluated against fungi and displayed
good fungicidal activities against Botrytis cinereal and Rhizoctonia solani. Preliminary …

Synthesis, fungicidal activity and molecular docking of novel pyrazole-carboxamides bearing a branched alkyl ether moiety

Q Xie, S Zhang, Y Zhang, B Zhang, F Wan, Y Li… - Bioorganic & Medicinal …, 2024 - Elsevier
Succinate dehydrogenase inhibitors are essential fungicides used in agriculture. To explore
new pyrazole-carboxamides with high fungicidal activity, a series of N-substitutedphenyl-3 …

Synthesis, fungicidal activity and SAR of 3, 4-dichloroisothiazole-based cycloalkylsulfonamides

Y Zhang, M Wang, M Ahmed, L He, M Ji, Z Qi… - Bioorganic & Medicinal …, 2019 - Elsevier
To develop more valuable and effective fungicide candidates, a novel series of 3, 4-
dichloroisothioxazole-based cycloalkylsulfonamides were synthesized and their structures …

N-(2-三氟甲基-4-氯苯基)-2-吡唑酰氨基环己烷基磺酰胺类化合物的合成与杀菌活性

孟司奇, 杨永贵, 纪明山, 祁之秋, 李兴海 - 农药学学报, 2018 - nyxxb.cn
吡唑酰胺类杀菌剂是近年新农药开发的热点. 本研究采用EDCI/HOBt 酰胺化法合成了14
个结构新颖的N-(2-三氟甲基-4-氯苯基)-2-吡唑酰氨基环己烷基磺酰胺类化合物(3a~ 3n) …

Synthesis, Fungicidal Activity and SAR of 2-Thiazolamide/Pyrazolamide-Cyclohexylsulfonamides against Botrytis cinerea

S Zhang, S Meng, Y Xie, Y Yang, Y Zhang, L He… - Molecules, 2019 - mdpi.com
In order to explore more efficient sulfonamides against Botrytis cinereal, 36 novel
cyclohexylsulfonamides were synthesized by N-(3-dimethylaminopropyl)-N …

吡啶联噁唑酰胺类化合物的设计, 合成及杀菌活性

陈澍, 任朝丽, 田晓雨, 张冬林, 杨森, 袁绍顷, 杜晓华… - 有机化学, 2021 - sioc-journal.cn
摘要以吡啶-2-甲醛为起始原料, 经环合, 氧化, 取代, 水解, 氯化和胺解反应, 采用中间体衍生化法
合成了13 个新型的吡啶联噁唑酰胺类化合物, 其结构经1H NMR 和高分辨质谱表征 …

Design, Synthesis and Fungicidal Activities of Pyridyl Oxazoamide Compounds

C Shu, R Chaoli, T Xiaoyu, Z Donglin, Y Sen… - Chinese Journal of …, 2021 - sioc-journal.cn
Thirteen novel pyridyl oxazoamide compounds were synthesized using pyridine-2-
formaldehyde as the starting material through cyclization, oxidation, substitution, hydrolysis …

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Y Zhang, M Wang, M Ahmed, L He, M Ji, Z Qi, X Li - 2019 - srcsignaling.com
To develop more valuable and effective fungicide candidates, a novel series of 3, 4-
dichloroisothioxazole-based cycloalkylsulfonamides were synthesized and their structures …